Global Patent Index - EP 1015453 A1

EP 1015453 A1 2000-07-05 - 3-(IODOPHENOXYMETHYL) CARBAPENEM ANTIBACTERIALS

Title (en)

3-(IODOPHENOXYMETHYL) CARBAPENEM ANTIBACTERIALS

Title (de)

ANTIBAKTERIELLE 3-(IODOPHENOXYMETHYL)CARBAPENEM

Title (fr)

ANTIBACTERIENS DU TYPE 3-(IODOPHENOXYMETHYL) CARBAPENEM

Publication

EP 1015453 A1 (EN)

Application

EP 98944779 A

Priority

  • GB 9815806 A
  • US 9818578 W
  • US 5822397 P

Abstract (en)

[origin: WO9912928A1] The present invention relates to carbapenem antibacterial agents in which the carbapenem nucleus is substituted at the 2-position with an iodo-substituted phenyl linked through a CH2-O- group. The compounds of the invention are represented by formula (I). Salts and hydrates thereof are included. The iodo-substituted phenyl ring is further substituted with various substituent groups including at least one cationic group. Pharmaceutical compositions and methods of treatment are also included.

IPC 1-7 (main, further and additional classification)

C07D 477/14; A61K 31/40

IPC 8 full level (invention and additional information)

C07D 487/08 (2006.01); A61K 31/397 (2006.01); A61K 31/407 (2006.01); A61K 31/4178 (2006.01); A61K 31/4439 (2006.01); A61K 31/499 (2006.01); A61P 31/04 (2006.01); C07D 477/00 (2006.01); C07D 477/14 (2006.01)

CPC (invention and additional information)

C07D 477/14 (2013.01)

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU NL PT SE

EPO simple patent family

WO 9912928 A1 19990318; AU 732335 B2 20010412; AU 9223698 A 19990329; CA 2302009 A1 19990318; EP 1015453 A1 20000705; EP 1015453 A4 20010919; JP 2003517427 A 20030527

INPADOC legal status


2002-10-23 [18D] DEEMED TO BE WITHDRAWN

- Effective date: 20020416

2002-01-23 [17Q] FIRST EXAMINATION REPORT

- Effective date: 20011205

2001-09-19 [A4] SUPPLEMENTARY SEARCH REPORT

- Effective date: 20010806

2001-09-19 [AK] DESIGNATED CONTRACTING STATES:

- Kind Code of Ref Document: A4

- Designated State(s): AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU NL PT SE

2001-09-19 [RIC1] CLASSIFICATION (CORRECTION)

- Free text: 7C 07D 477/14 A, 7A 61K 31/40 B, 7C 07D 519/00 B, 7A 61K 31/495 B

2000-07-05 [17P] REQUEST FOR EXAMINATION FILED

- Effective date: 20000410

2000-07-05 [AK] DESIGNATED CONTRACTING STATES:

- Kind Code of Ref Document: A1

- Designated State(s): AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU NL PT SE

2000-07-05 [AX] REQUEST FOR EXTENSION OF THE EUROPEAN PATENT TO

- Free text: AL PAYMENT 20000410;LT PAYMENT 20000410;LV PAYMENT 20000410;MK PAYMENT 20000410;RO PAYMENT 20000410;SI PAYMENT 20000410