Global Patent Index - EP 1015454 A1

EP 1015454 A1 2000-07-05 - METHOD OF INHIBITING SERINE PROTEASE ENZYMES

Title (en)

METHOD OF INHIBITING SERINE PROTEASE ENZYMES

Title (de)

VERFAHREN ZUR VERHINDERUNG DER AKTIVITÄT DES SERINE PROTEASENZYMS

Title (fr)

PROCEDE D'INHIBITION D'ENZYMES SERINE PROTEASES

Publication

EP 1015454 A1 (EN)

Application

EP 98948907 A

Priority

  • EP 9805607 W
  • GB 9719189 A

Abstract (en)

[origin: WO9912932A1] According to the invention there is provided an inhibitor of a serine protease enzyme which is a substituted derivative of trans-hexahydropyrrolo[3,2-b]pyrrol-2-one save that it is not a compound of formula IA and IB (as defined in Annex 1).

IPC 1-7 (main, further and additional classification)

C07D 487/04; A61K 31/40

IPC 8 full level (invention and additional information)

G01N 33/50 (2006.01); A61K 31/407 (2006.01); A61P 7/02 (2006.01); A61P 11/00 (2006.01); A61P 11/06 (2006.01); A61P 31/22 (2006.01); A61P 43/00 (2006.01); C07B 61/00 (2006.01); C07D 207/14 (2006.01); C07D 487/04 (2006.01); G01N 33/15 (2006.01)

CPC (invention and additional information)

C07D 487/04 (2013.01); C07D 207/14 (2013.01)

Citation (search report)

See references of WO 9912932A1

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

EPO simple patent family

WO 9912932 A1 19990318; AU 9536298 A 19990329; EP 1015454 A1 20000705; GB 9719189 D0 19971112; JP 2001515903 A 20010925; ZA 9808160 B 20000322

INPADOC legal status


2003-10-08 [18D] DEEMED TO BE WITHDRAWN

- Effective date: 20030409

2003-01-08 [17Q] FIRST EXAMINATION REPORT

- Effective date: 20021126

2000-07-05 [17P] REQUEST FOR EXAMINATION FILED

- Effective date: 20000301

2000-07-05 [AK] DESIGNATED CONTRACTING STATES:

- Kind Code of Ref Document: A1

- Designated State(s): AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE