EP 1015454 A1 20000705 - METHOD OF INHIBITING SERINE PROTEASE ENZYMES
Title (en)
METHOD OF INHIBITING SERINE PROTEASE ENZYMES
Title (de)
VERFAHREN ZUR VERHINDERUNG DER AKTIVITÄT DES SERINE PROTEASENZYMS
Title (fr)
PROCEDE D'INHIBITION D'ENZYMES SERINE PROTEASES
Publication
Application
Priority
- EP 9805607 W 19980907
- GB 9719189 A 19970909
Abstract (en)
[origin: WO9912932A1] According to the invention there is provided an inhibitor of a serine protease enzyme which is a substituted derivative of trans-hexahydropyrrolo[3,2-b]pyrrol-2-one save that it is not a compound of formula IA and IB (as defined in Annex 1).
IPC 1-7
IPC 8 full level
A61K 31/407 (2006.01); A61P 7/02 (2006.01); A61P 11/00 (2006.01); A61P 11/06 (2006.01); A61P 31/22 (2006.01); A61P 43/00 (2006.01); C07B 61/00 (2006.01); C07D 207/14 (2006.01); C07D 487/04 (2006.01); G01N 33/15 (2006.01); G01N 33/50 (2006.01)
CPC (source: EP)
A61P 7/02 (2017.12); A61P 11/00 (2017.12); A61P 11/06 (2017.12); A61P 31/22 (2017.12); A61P 43/00 (2017.12); C07D 207/14 (2013.01); C07D 487/04 (2013.01)
Citation (search report)
See references of WO 9912932A1
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
WO 9912932 A1 19990318; AU 9536298 A 19990329; EP 1015454 A1 20000705; GB 9719189 D0 19971112; JP 2001515903 A 20010925; ZA 988160 B 20000322
DOCDB simple family (application)
EP 9805607 W 19980907; AU 9536298 A 19980907; EP 98948907 A 19980907; GB 9719189 A 19970909; JP 2000510739 A 19980907; ZA 988160 A 19980907