Global Patent Index - EP 1017393 A1

EP 1017393 A1 20000712 - PYRAZINONE THROMBIN INHIBITORS

Title (en)

PYRAZINONE THROMBIN INHIBITORS

Title (de)

PYRAZINON THROMBININHIBITOREN

Title (fr)

INHIBITEURS DE THROMBINE A BASE DE PYRAZINONE

Publication

EP 1017393 A1 20000712 (EN)

Application

EP 98946835 A 19980903

Priority

  • GB 9801005 A 19980116
  • US 9818417 W 19980903
  • US 5805897 P 19970905

Abstract (en)

[origin: WO9911267A1] Compounds of the invention are useful in inhibiting thrombin and associated thrombotic occlusions having structure (a), for example, structure (17-1).

IPC 1-7

A61K 31/495; C07D 241/20; C07D 401/12; C07D 401/14; C07D 405/12; C07D 405/14

IPC 8 full level

C07D 241/20 (2006.01); A61K 31/4965 (2006.01); A61K 31/497 (2006.01); A61P 7/02 (2006.01); C07D 401/12 (2006.01); C07D 401/14 (2006.01); C07D 405/12 (2006.01); C07D 405/14 (2006.01)

CPC (source: EP)

A61P 7/02 (2017.12); C07D 401/12 (2013.01); C07D 401/14 (2013.01); C07D 405/14 (2013.01)

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU NL PT SE

DOCDB simple family (publication)

WO 9911267 A1 19990311; CA 2301520 A1 19990311; EP 1017393 A1 20000712; EP 1017393 A4 20020123; JP 2001514227 A 20010911

DOCDB simple family (application)

US 9818417 W 19980903; CA 2301520 A 19980903; EP 98946835 A 19980903; JP 2000508369 A 19980903