EP 1017393 A4 20020123 - PYRAZINONE THROMBIN INHIBITORS
Title (en)
PYRAZINONE THROMBIN INHIBITORS
Title (de)
PYRAZINON THROMBININHIBITOREN
Title (fr)
INHIBITEURS DE THROMBINE A BASE DE PYRAZINONE
Publication
Application
Priority
- GB 9801005 A 19980116
- US 9818417 W 19980903
- US 5805897 P 19970905
Abstract (en)
[origin: WO9911267A1] Compounds of the invention are useful in inhibiting thrombin and associated thrombotic occlusions having structure (a), for example, structure (17-1).
IPC 1-7
IPC 8 full level
C07D 241/20 (2006.01); A61K 31/4965 (2006.01); A61K 31/497 (2006.01); A61P 7/02 (2006.01); C07D 401/12 (2006.01); C07D 401/14 (2006.01); C07D 405/12 (2006.01); C07D 405/14 (2006.01)
CPC (source: EP)
A61P 7/02 (2018.01); C07D 401/12 (2013.01); C07D 401/14 (2013.01); C07D 405/14 (2013.01)
Citation (search report)
[X] WO 9701338 A1 19970116 - MERCK & CO INC [US], et al
Citation (examination)
- SANDERSON et al. "Small, Noncovalent Serine Protease Inhibitors" MEDICINAL RESEARCH REVIEWS, 1999, VOL 19, NR 2, 179-197
- See also references of WO 9911267A1
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU NL PT SE
DOCDB simple family (publication)
WO 9911267 A1 19990311; CA 2301520 A1 19990311; EP 1017393 A1 20000712; EP 1017393 A4 20020123; JP 2001514227 A 20010911
DOCDB simple family (application)
US 9818417 W 19980903; CA 2301520 A 19980903; EP 98946835 A 19980903; JP 2000508369 A 19980903