Global Patent Index - EP 1020446 A1

EP 1020446 A1 2000-07-19 - NAPHTHALIMIDOBENZAMIDE DERIVATIVES

Title (en)

NAPHTHALIMIDOBENZAMIDE DERIVATIVES

Title (de)

NAPHTHIMIDOBENZAMID-DERIVATE

Title (fr)

DERIVES DE NAPHTALIMIDOBENZAMIDE

Publication

EP 1020446 A1 (EN)

Application

EP 99926895 A

Priority

  • JP 9903574 W
  • JP 18907898 A

Abstract (en)

The present invention relates to a naphthalimidobenzamide derivative represented by the following formula (1): <CHEM> (wherein, R<1> represents a hydrogen atom, etc., Y represents a hydrogen atom or -CON(R<4>)-A<2>-X<2>, R<2> and R<4> are the same or different and each independently represents a hydrogen atom, etc., A<1> and A<2> are the same or different and each independently represents an alkylene group which may be interrupted at least once by -N(R<3>)- (R<3> representing a hydrogen atom, etc.) and X<1> and X<2> are the same or different and each independently represents a (hetero)aryl group which may have a substituent, etc.) or salt thereof; and a pharmaceutical comprising it as an effective ingredient. The compound is useful as an antitumor agent and the like.

IPC 1-7 (main, further and additional classification)

C07D 221/14; A61K 31/47; A61K 31/495; A61K 31/535; C07D 401/12; C07D 401/14

IPC 8 full level (invention and additional information)

C07D 221/14 (2006.01); C07D 401/14 (2006.01); C07D 471/04 (2006.01); C07D 519/00 (2006.01)

CPC (invention and additional information)

C07D 221/14 (2013.01); C07D 401/14 (2013.01); C07D 471/04 (2013.01)

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

DOCDB simple family

EP 1020446 A1 20000719; EP 1020446 A4 20011107; EP 1020446 B1 20060315; AT 320417 T 20060415; AU 4396399 A 20000124; AU 727591 B2 20001214; CA 2300069 A1 20000113; CA 2300069 C 20060117; DE 69930383 D1 20060511; DE 69930383 T2 20061005; JP 3357662 B2 20021216; KR 100364205 B1 20021211; KR 20010023464 A 20010326; US 6300331 B1 20011009; WO 0001672 A1 20000113