Global Patent Index - EP 1021436 A1

EP 1021436 A1 20000726 - ETHYL 4-(8-CHLORO-5, 6-DIHYDRO-11H- BENZO 5,6 CYCLOHEPTA 1,2-b PYRIDIN -11-YLIDENE)-1- PIPERIDENE CARBOXYLATE POLYMORPH

Title (en)

ETHYL 4-(8-CHLORO-5, 6-DIHYDRO-11H- BENZO 5,6 CYCLOHEPTA 1,2-b PYRIDIN -11-YLIDENE)-1- PIPERIDENE CARBOXYLATE POLYMORPH

Title (de)

ETHYL4-(8-CHLORO-5,6-DIHYDRO-11H-BENZO¬5,6 CYCCLOHEPTA¬1,2 PYRIDIN-11-YLIDENE)-1-PIPERIDENCARBOXYLATPOLYMORPPH

Title (fr)

POLYMORPHE D'ETHYL 4-(8-CHLORO-5, 6,-DIHYDRO-11H- BENZO 5,6 CYCLOHEPTA 1,2-b PYRIDINE -11-YLIDENE)-1- PIPERIDENE CARBOXYLATE

Publication

EP 1021436 A1 20000726 (EN)

Application

EP 98950916 A 19981008

Priority

  • US 9820919 W 19981008
  • US 94888697 A 19971010

Abstract (en)

[origin: WO9919322A1] A polymorph form 2 of ethyl 4-(8-chloro-5, 6-dihydro-11H- benzo[5,6]cyclohepta [1,2-b]pyridin -11-ylidene)-1- piperidene carboxylate (hereinafter "loratadine") represented by formula (I). Pharmaceutical composition containing the polymorph form 2, and methods of using the polymorph form 2 to treat allergic reactions in mammals such as man are disclosed.

IPC 1-7

C07D 401/04; A61K 31/445

IPC 8 full level

A61K 31/4427 (2006.01); A61K 31/4545 (2006.01); A61P 37/08 (2006.01); C07D 401/04 (2006.01)

CPC (source: EP)

A61P 37/08 (2017.12); C07D 401/04 (2013.01)

Citation (search report)

See references of WO 9919322A1

Designated contracting state (EPC)

AT BE CH DE DK ES FI FR GB GR IE IT LI LU NL PT SE

Designated extension state (EPC)

LT LV RO

DOCDB simple family (publication)

WO 9919322 A1 19990422; AU 9683798 A 19990503; CA 2305801 A1 19990422; EP 1021436 A1 20000726; JP 2001519428 A 20011023

DOCDB simple family (application)

US 9820919 W 19981008; AU 9683798 A 19981008; CA 2305801 A 19981008; EP 98950916 A 19981008; JP 2000515894 A 19981008