Global Patent Index - EP 1023268 A1

EP 1023268 A1 2000-08-02 - ISOQUINOLINES AS UROKINASE INHIBITORS

Title (en)

ISOQUINOLINES AS UROKINASE INHIBITORS

Title (de)

ISOCHINOLIN DERIVATE ALS UROKINASE INHIBITOREN

Title (fr)

ISOQUINOLINES EN TANT QU'INHIBITEURS DE L'UROKINASE

Publication

EP 1023268 A1 (EN)

Application

EP 98954357 A

Priority

  • EP 9806353 W
  • GB 9721964 A

Abstract (en)

[origin: WO9920608A1] Compounds of formula (I) and pharmaceutically acceptable salts thereof, wherein one of R<1> and R<2> is H and the other is N=C(NH2)2 or NHC(=NH)NH2, and the other substituents are as defined herein, are urokinase (uPA) inhibitors.

IPC 1-7 (main, further and additional classification)

C07D 217/22; A61K 31/47; C07D 401/06; C07D 405/04; C07D 409/04; C07D 491/04

IPC 8 full level (invention and additional information)

A61K 31/472 (2006.01); A61K 31/4725 (2006.01); A61K 31/4741 (2006.01); A61K 31/497 (2006.01); A61K 31/5377 (2006.01); A61P 15/08 (2006.01); A61P 17/02 (2006.01); A61P 19/00 (2006.01); A61P 19/02 (2006.01); A61P 29/00 (2006.01); A61P 35/04 (2006.01); A61P 43/00 (2006.01); C07D 217/22 (2006.01); C07D 217/24 (2006.01); C07D 401/04 (2006.01); C07D 401/06 (2006.01); C07D 401/12 (2006.01); C07D 405/04 (2006.01); C07D 409/04 (2006.01); C07D 491/04 (2006.01); C07D 491/056 (2006.01); C07D 521/00 (2006.01)

CPC (invention and additional information)

C07D 231/12 (2013.01); C07D 217/22 (2013.01); C07D 233/56 (2013.01); C07D 249/08 (2013.01); C07D 401/04 (2013.01); C07D 405/04 (2013.01); C07D 409/04 (2013.01); C07D 491/04 (2013.01)

Citation (search report)

See references of WO 9920608A1

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU NL PT SE

EPO simple patent family

WO 9920608 A1 19990429; AP 959 A 20010417; AP 9801366 A0 19981231; AR 015964 A1 20010530; AT 240943 T 20030615; AU 1150899 A 19990510; AU 727315 B2 20001207; BG 104328 A 20001229; BR 9812922 A 20000808; CA 2306782 A1 19990429; CA 2306782 C 20050517; CN 1275979 A 20001206; CO 4990959 A1 20001226; DE 69814894 D1 20030626; DE 69814894 T2 20031224; DK 1023268 T3 20030610; DZ 2624 A1 20030308; EA 002632 B1 20020829; EA 200000320 A1 20001030; EP 1023268 A1 20000802; EP 1023268 B1 20030521; ES 2197514 T3 20040101; GB 9721964 D0 19971217; GT 199800159 A 20000401; HN 1998000158 A 19990209; HR P20000217 A2 20001031; HU 0004491 A2 20010328; HU 0004491 A3 20021028; ID 23913 A 20000525; IL 135122 D0 20010520; IS 5412 A 20000321; JP 2001520221 A 20011030; JP 3600794 B2 20041215; KR 20010031163 A 20010416; MA 26552 A1 20041220; NO 20001924 A 20000615; NO 20001924 D0 20000413; NZ 503390 A 20020328; OA 11348 A 20031218; PA 8461601 A1 20000524; PE 121299 A1 19991201; PL 340035 A1 20010115; PT 1023268 E 20030930; SK 4872000 A3 20011203; TN SN98185 A1 20050315; TR 200001010 T2 20000921; US 6248738 B1 20010619; UY 25211 A1 20001229; YU 21100 A 20021115; ZA 9809412 B 20000417

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