EP 1025090 A4 20001108 - VITRONECTIN RECEPTOR ANTAGONISTS
Title (en)
VITRONECTIN RECEPTOR ANTAGONISTS
Title (de)
VITRONECTIN-REZEPTOR-ANTAGONISTEN
Title (fr)
ANTAGONISTES DU RECEPTEUR DE LA VITRONECTINE
Publication
Application
Priority
- US 9819466 W 19980918
- US 5934297 P 19970919
- US 6343897 P 19971029
Abstract (en)
[origin: WO9915508A1] Compounds of formula (I) are disclosed which are vitronectin receptor antagonists and are useful in the treatment of osteoporosis wherein: A is CH2 or O; R<1> is H, halo or C1-6alkyl; R<2> is H, C1-6alkyl or CH2NR''R''; X is O or CH2; Y is (a), (b), (c), (d), (e), (f) or (g); G is NR'', S or O; R' is H, C1-6alkyl, OC1-6alkyl, SC1-6alkyl, NR''R'' or halo; each R'' independently is H or C1-6alkyl; and s is 0, 1 or 2; or a pharmaceutically acceptable salt thereof.
IPC 1-7
C07D 213/74; A61K 31/44; C07D 213/73; C07D 217/22; C07D 239/14; C07D 277/42; C07D 405/12
IPC 8 full level
A61K 31/426 (2006.01); A61K 31/44 (2006.01); A61K 31/4418 (2006.01); A61K 31/4427 (2006.01); A61K 31/443 (2006.01); A61K 31/47 (2006.01); A61K 31/472 (2006.01); C07D 239/02 (2006.01); A61K 31/505 (2006.01); A61K 31/506 (2006.01); A61P 9/00 (2006.01); A61P 9/10 (2006.01); A61P 19/10 (2006.01); A61P 29/00 (2006.01); A61P 35/00 (2006.01); A61P 35/04 (2006.01); A61P 43/00 (2006.01); C07D 213/73 (2006.01); C07D 213/74 (2006.01); C07D 217/12 (2006.01); C07D 217/22 (2006.01); C07D 239/14 (2006.01); C07D 277/20 (2006.01); C07D 277/38 (2006.01); C07D 277/42 (2006.01); C07D 405/12 (2006.01)
CPC (source: EP KR)
A61P 9/00 (2018.01 - EP); A61P 9/10 (2018.01 - EP); A61P 19/10 (2018.01 - EP); A61P 29/00 (2018.01 - EP); A61P 35/00 (2018.01 - EP); A61P 35/04 (2018.01 - EP); A61P 43/00 (2018.01 - EP); C07D 213/73 (2013.01 - EP KR); C07D 213/74 (2013.01 - EP KR); C07D 217/22 (2013.01 - EP KR); C07D 233/48 (2013.01 - KR); C07D 239/14 (2013.01 - EP KR); C07D 263/58 (2013.01 - KR); C07D 277/42 (2013.01 - EP KR); C07D 313/14 (2013.01 - KR); C07D 405/06 (2013.01 - KR); C07D 405/12 (2013.01 - EP KR); C07D 487/04 (2013.01 - KR)
Citation (search report)
- [X] WO 9701540 A1 19970116 - SMITHKLINE BEECHAM CORP [US], et al
- [PX] WO 9830542 A1 19980716 - SMITHKLINE BEECHAM CORP [US], et al
- [PX] WO 9815278 A1 19980416 - SMITHKLINE BEECHAM CORP [US], et al
- See also references of WO 9915508A1
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
WO 9915508 A1 19990401; AP 2000001766 A0 19980918; AR 015446 A1 20010502; AU 738433 B2 20010920; AU 9397298 A 19990412; BG 104314 A 20010131; BR 9812340 A 20011218; CA 2303487 A1 19990401; CN 1278250 A 20001227; CO 5011087 A1 20010228; DZ 2609 A1 20030301; EA 200000336 A1 20001030; EP 1025090 A1 20000809; EP 1025090 A4 20001108; HU P0003641 A2 20010328; HU P0003641 A3 20021028; ID 24162 A 20000713; IL 135028 A0 20010520; JP 2001517658 A 20011009; KR 20010024141 A 20010326; MA 26547 A1 20041220; NO 20001407 D0 20000317; NO 20001407 L 20000317; NZ 503389 A 20020328; OA 11341 A 20031210; PE 122699 A1 20000212; PL 339381 A1 20001218; SK 4082000 A3 20000912; TR 200000721 T2 20001121; TW 513303 B 20021211
DOCDB simple family (application)
US 9819466 W 19980918; AP 2000001766 A 19980918; AR P980104604 A 19980916; AU 9397298 A 19980918; BG 10431400 A 20000407; BR 9812340 A 19980918; CA 2303487 A 19980918; CN 98810811 A 19980918; CO 98053986 A 19980918; DZ 980219 A 19980916; EA 200000336 A 19980918; EP 98947116 A 19980918; HU P0003641 A 19980918; ID 20000468 A 19980918; IL 13502898 A 19980918; JP 2000512816 A 19980918; KR 20007002901 A 20000318; MA 25266 A 19980918; NO 20001407 A 20000317; NZ 50338998 A 19980918; OA 1200000079 A 20000316; PE 00088198 A 19980916; PL 33938198 A 19980918; SK 4082000 A 19980918; TR 200000721 T 19980918; TW 87115535 A 19980923