Global patent index - EP 1027042 A1

EP 1027042 A1 2000-08-16 - INHIBITORS OF FARNESYL PROTEIN TRANSFERASE

Title (en)

INHIBITORS OF FARNESYL PROTEIN TRANSFERASE

Title (de)

INHIBITOREN DER FARNESYL PROTEIN TRANSFERASE

Title (fr)

INHIBITEURS DE LA TRANSFERASE FARNESYLE PROTEINE

Publication

EP 1027042 A1 (EN)

Application

EP 98948279 A

Priority

  • US 9819315 W
  • US 6082397 P

Abstract (en)

[origin: WO9918951A1] Inhibition of farnesyl transferase, which is an enzyme involved in ras oncogene expression, is effected by compounds of formulas (I), (II), their enantiomers, diastereomers, and pharmaceutically acceptable salts, prodrugs and solvates thereof inhibit farnesyl protein transferase which is an enzyme involved in ras oncogene expression.

IPC 1-7 (main, further and additional classification)

A61K 31/33; A61K 31/495; A61K 31/50; A61K 31/53; A61K 31/535; A61K 31/54; A61K 31/55; A61P 35/00; C07D 237/26; C07D 239/70; C07D 241/36; C07D 243/12; C07D 243/14; C07D 401/06; C07D 401/12; C07D 403/06; C07D 403/12; C07D 409/06

IPC 8 full level (invention and additional information)

A61K 31/551 (2006.01); A61K 31/5513 (2006.01); A61P 35/00 (2006.01); A61P 43/00 (2006.01); C07D 243/12 (2006.01); C07D 243/14 (2006.01); C07D 401/06 (2006.01); C07D 401/12 (2006.01); C07D 403/06 (2006.01); C07D 403/12 (2006.01); C07D 409/06 (2006.01)

CPC (invention and additional information)

C07D 401/06 (2013.01); C07D 243/14 (2013.01); C07D 401/12 (2013.01); C07D 403/06 (2013.01); C07D 403/12 (2013.01); C07D 409/06 (2013.01)

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

EPO simple patent family

WO 9918951 A1 19990422; AU 735366 B2 20010705; AU 9488698 A 19990503; CA 2304473 A1 19990422; EP 1027042 A1 20000816; EP 1027042 A4 20040818; JP 2001519387 A 20011023

INPADOC legal status

2006-10-04 [18D] DEEMED TO BE WITHDRAWN

- Ref Legal Event Code: 18D

- Effective date: 20060331

2004-08-18 [A4] SUPPLEMENTARY SEARCH REPORT

- Ref Legal Event Code: A4

- Effective date: 20040706

2004-08-18 [RIC1] CLASSIFICATION (CORRECTION)

- Ref Legal Event Code: RIC1

- IPC: 7A 61K 31/33 A

2004-08-18 [RIC1] CLASSIFICATION (CORRECTION)

- Ref Legal Event Code: RIC1

- IPC: 7A 61K 31/495 B

2004-08-18 [RIC1] CLASSIFICATION (CORRECTION)

- Ref Legal Event Code: RIC1

- IPC: 7A 61K 31/50 B

2004-08-18 [RIC1] CLASSIFICATION (CORRECTION)

- Ref Legal Event Code: RIC1

- IPC: 7A 61K 31/53 B

2004-08-18 [RIC1] CLASSIFICATION (CORRECTION)

- Ref Legal Event Code: RIC1

- IPC: 7A 61K 31/535 B

2004-08-18 [RIC1] CLASSIFICATION (CORRECTION)

- Ref Legal Event Code: RIC1

- IPC: 7A 61K 31/54 B

2004-08-18 [RIC1] CLASSIFICATION (CORRECTION)

- Ref Legal Event Code: RIC1

- IPC: 7A 61K 31/55 B

2004-08-18 [RIC1] CLASSIFICATION (CORRECTION)

- Ref Legal Event Code: RIC1

- IPC: 7C 07D 237/26 B

2004-08-18 [RIC1] CLASSIFICATION (CORRECTION)

- Ref Legal Event Code: RIC1

- IPC: 7C 07D 239/70 B

2004-08-18 [RIC1] CLASSIFICATION (CORRECTION)

- Ref Legal Event Code: RIC1

- IPC: 7C 07D 241/36 B

2004-08-18 [RIC1] CLASSIFICATION (CORRECTION)

- Ref Legal Event Code: RIC1

- IPC: 7C 07D 243/12 B

2004-08-18 [RIC1] CLASSIFICATION (CORRECTION)

- Ref Legal Event Code: RIC1

- IPC: 7C 07D 243/14 B

2004-08-18 [RIC1] CLASSIFICATION (CORRECTION)

- Ref Legal Event Code: RIC1

- IPC: 7C 07D 401/06 B

2004-08-18 [RIC1] CLASSIFICATION (CORRECTION)

- Ref Legal Event Code: RIC1

- IPC: 7C 07D 409/06 B

2004-08-18 [RIC1] CLASSIFICATION (CORRECTION)

- Ref Legal Event Code: RIC1

- IPC: 7C 07D 401/12 B

2004-08-18 [RIC1] CLASSIFICATION (CORRECTION)

- Ref Legal Event Code: RIC1

- IPC: 7C 07D 403/12 B

2004-08-18 [RIC1] CLASSIFICATION (CORRECTION)

- Ref Legal Event Code: RIC1

- IPC: 7C 07D 403/06 B

2004-08-18 [RIC1] CLASSIFICATION (CORRECTION)

- Ref Legal Event Code: RIC1

- IPC: 7A 61P 35/00 B

2000-08-16 [17P] REQUEST FOR EXAMINATION FILED

- Ref Legal Event Code: 17P

- Effective date: 20000427

2000-08-16 [AK] DESIGNATED CONTRACTING STATES:

- Ref Legal Event Code: AK

- Designated State(s): AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE