EP 1027042 A1 20000816 - INHIBITORS OF FARNESYL PROTEIN TRANSFERASE
Title (en)
INHIBITORS OF FARNESYL PROTEIN TRANSFERASE
Title (de)
INHIBITOREN DER FARNESYL PROTEIN TRANSFERASE
Title (fr)
INHIBITEURS DE LA TRANSFERASE FARNESYLE PROTEINE
Publication
Application
Priority
- US 9819315 W 19980916
- US 6082397 P 19970929
Abstract (en)
[origin: WO9918951A1] Inhibition of farnesyl transferase, which is an enzyme involved in ras oncogene expression, is effected by compounds of formulas (I), (II), their enantiomers, diastereomers, and pharmaceutically acceptable salts, prodrugs and solvates thereof inhibit farnesyl protein transferase which is an enzyme involved in ras oncogene expression.
IPC 1-7
A61K 31/33; A61K 31/495; A61K 31/50; A61K 31/53; A61K 31/535; A61K 31/54; A61K 31/55; C07D 237/26; C07D 239/70; C07D 241/36; C07D 243/12; C07D 243/14; C07D 401/06; C07D 409/06; C07D 401/12; C07D 403/12; C07D 403/06; A61P 35/00
IPC 8 full level
A61K 31/551 (2006.01); A61K 31/5513 (2006.01); A61P 35/00 (2006.01); A61P 43/00 (2006.01); C07D 243/12 (2006.01); C07D 243/14 (2006.01); C07D 401/06 (2006.01); C07D 401/12 (2006.01); C07D 403/06 (2006.01); C07D 403/12 (2006.01); C07D 409/06 (2006.01)
CPC (source: EP)
A61P 35/00 (2017.12); A61P 43/00 (2017.12); C07D 243/14 (2013.01); C07D 401/06 (2013.01); C07D 401/12 (2013.01); C07D 403/06 (2013.01); C07D 403/12 (2013.01); C07D 409/06 (2013.01)
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
WO 9918951 A1 19990422; AU 735366 B2 20010705; AU 9488698 A 19990503; CA 2304473 A1 19990422; EP 1027042 A1 20000816; EP 1027042 A4 20040818; JP 2001519387 A 20011023
DOCDB simple family (application)
US 9819315 W 19980916; AU 9488698 A 19980916; CA 2304473 A 19980916; EP 98948279 A 19980916; JP 2000515586 A 19980916