EP 1027046 A4 20020403 - ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE

Title (en)

ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE

Title (de)

ANTAGONISTEN DES GONADOTROPIN FREISETZENDEN HORMONS

Title (fr)

ANTAGONISTES DE L'HORMONE DE LIBERATION DE LA GONADOTHROPHINE

Publication

EP 1027046 A4 20020403 (EN)

Application

EP 98954019 A 19981027

Priority

GB 9809789 A 19980507
US 9822799 W 19981027
US 6330597 P 19971028

Abstract (en)

[origin: WO9921553A1] There are disclosed compounds of formula (I) and pharmaceutically acceptable salts thereof which are useful as antagonists of GnRH and as such may be useful for the treatment of a variety of sex-hormone related and other conditions in both men and women.

IPC 1-7

A61K 31/405; A61K 31/35; C07D 209/04; C07D 209/14; C07D 209/42; A61P 5/24; C07D 453/06; C07D 487/08

IPC 8 full level

A61K 31/403 (2006.01); A61K 31/404 (2006.01); A61K 31/4045 (2006.01); A61K 31/454 (2006.01); A61K 31/513 (2006.01); A61K 31/5377 (2006.01); A61P 1/04 (2006.01); A61P 11/00 (2006.01); A61P 15/00 (2006.01); A61P 15/18 (2006.01); A61P 17/00 (2006.01); A61P 25/20 (2006.01); A61P 35/00 (2006.01); A61P 43/00 (2006.01); C07D 209/14 (2006.01); C07D 453/06 (2006.01); C07D 487/08 (2006.01)

CPC (source: EP)

A61P 1/04 (2017.12); A61P 5/24 (2017.12); A61P 11/00 (2017.12); A61P 15/00 (2017.12); A61P 15/18 (2017.12); A61P 17/00 (2017.12); A61P 25/20 (2017.12); A61P 35/00 (2017.12); A61P 43/00 (2017.12); C07D 453/06 (2013.01); C07D 487/08 (2013.01)

Citation (search report)

[X] FR 2181559 A1 19731207 - AEC CHIMIE ORGANIQUE BIO [FR]
[X] GB 1562825 A 19800319 - LILLY CO ELI
[XD] US 5030640 A 19910709 - FISHER MICHAEL H [US], et al
[XD] US 4544663 A 19851001 - MANNING ROBERT E [US], et al
[E] WO 9855119 A1 19981210 - MERCK & CO INC [US], et al
See references of WO 9921553A1

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU NL PT SE

DOCDB simple family (publication)

WO 9921553 A1 19990506; AU 1124399 A 19990517; CA 2308454 A1 19990506; EP 1027046 A1 20000816; EP 1027046 A4 20020403; JP 2001520996 A 20011106

DOCDB simple family (application)

US 9822799 W 19981027; AU 1124399 A 19981027; CA 2308454 A 19981027; EP 98954019 A 19981027; JP 2000517711 A 19981027