Global Patent Index - EP 1027352 A1

EP 1027352 A1 2000-08-16 - CARBAPENEM ANTIBACTERIAL COMPOUNDS, COMPOSITIONS AND METHODS OF TREATMENT

Title (en)

CARBAPENEM ANTIBACTERIAL COMPOUNDS, COMPOSITIONS AND METHODS OF TREATMENT

Title (de)

ANTIBAKTERIELLE CARBAPENEM-VERBINDUNGEN, ZUSAMMENSETZUNGEN UND BEHANDLUNGSMETHODEN

Title (fr)

COMPOSES ANTIBACTERIENS DE LA CLASSE DES CARBAPENEMES, COMPOSITIONS ET PROCEDES DE TRAITEMENT

Publication

EP 1027352 A1 (EN)

Application

EP 98953736 A

Priority

  • GB 9806431 A
  • US 9822110 W
  • US 6303197 P

Abstract (en)

[origin: WO9920627A1] Compounds of formula (I) are disclosed as well as pharmaceutically acceptable salts thereof. The naphthosultam is substituted with various substituent groups including at least one cationic group -A-Q-L-B. The carbapenems of the invention are effective against susceptible bacterial organisms, including methicillin resistant Staphylococcus aureus (MRSA), methicillin resistant Staphylococcus epidermidis (MRSE), and methicillin resistant coagulase negative Staphylococci (MRCNS).

IPC 1-7 (main, further and additional classification)

C07D 477/14; A61K 31/495; A61K 31/55

IPC 8 full level (invention and additional information)

C07D 477/00 (2006.01); A61K 31/397 (2006.01); A61K 31/496 (2006.01); A61K 31/506 (2006.01); A61P 31/04 (2006.01); C07D 477/14 (2006.01)

CPC (invention and additional information)

C07D 477/14 (2013.01)

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU NL PT SE

EPO simple patent family

WO 9920627 A1 19990429; AU 1103099 A 19990510; AU 739799 B2 20011018; CA 2306565 A1 19990429; EP 1027352 A1 20000816; EP 1027352 A4 20010919; JP 2002509856 A 20020402

INPADOC legal status


2004-07-14 [18D] DEEMED TO BE WITHDRAWN

- Ref Legal Event Code: 18D

- Effective date: 20040108

2002-01-16 [17Q] FIRST EXAMINATION REPORT

- Ref Legal Event Code: 17Q

- Effective date: 20011204

2001-09-19 [A4] SUPPLEMENTARY SEARCH REPORT

- Ref Legal Event Code: A4

- Effective date: 20010807

2001-09-19 [AK] DESIGNATED CONTRACTING STATES:

- Ref Legal Event Code: AK

- Designated State(s): AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU NL PT SE

2001-09-19 [RIC1] CLASSIFICATION (CORRECTION)

- Ref Legal Event Code: RIC1

- Free Format Text: 7C 07D 477/14 A, 7A 61K 31/55 B, 7A 61K 31/495 B, 7C 07D 519/00 B

2000-08-16 [17P] REQUEST FOR EXAMINATION FILED

- Ref Legal Event Code: 17P

- Effective date: 20000523

2000-08-16 [AK] DESIGNATED CONTRACTING STATES:

- Ref Legal Event Code: AK

- Designated State(s): AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU NL PT SE

2000-08-16 [AX] REQUEST FOR EXTENSION OF THE EUROPEAN PATENT TO

- Ref Legal Event Code: AX

- Free Format Text: AL PAYMENT 20000523;LT PAYMENT 20000523;LV PAYMENT 20000523;MK PAYMENT 20000523;RO PAYMENT 20000523;SI PAYMENT 20000523