Global Patent Index - EP 1030844 A1

EP 1030844 A1 20000830 - COMPOUNDS WHICH INHIBIT TRYPTASE ACTIVITY

Title (en)

COMPOUNDS WHICH INHIBIT TRYPTASE ACTIVITY

Title (de)

VERBINDUNGEN, DIE DIE AKTIVITÄT VON TRYPTASE HEMMEN

Title (fr)

COMPOSES INHIBANT L'ACTIVITE DE LA TRYPTASE

Publication

EP 1030844 A1 20000830 (EN)

Application

EP 98955238 A 19981103

Priority

  • US 9823362 W 19981103
  • US 6515497 P 19971110
  • US 17969598 A 19981027

Abstract (en)

[origin: WO9924407A1] The present invention is directed to compounds which are capable of inhibiting the activity of tryptase. Such compounds are useful in the treatment or prevention of inflammatory disease, particularly those disease states which are mediated by mast cell activation. Also encompassed by the invention are formulations comprising the noted compounds, processes for preparing such compounds and methods for treating or preventing an inflammatory disease.

IPC 1-7

C07D 235/16; C07D 209/18; C07D 209/42; C07D 333/60; C07D 333/62; C07D 235/14; C07D 209/08; C07D 401/12; C07D 403/12; C07D 409/12; C07C 257/18; A61K 31/155; A61K 31/40; A61K 31/415; A61K 31/38

IPC 8 full level

C07C 257/18 (2006.01); C07D 209/08 (2006.01); C07D 235/16 (2006.01); C07D 235/20 (2006.01); C07D 333/08 (2006.01); C07D 401/12 (2006.01); C07D 409/12 (2006.01)

CPC (source: EP)

C07C 257/18 (2013.01); C07D 209/08 (2013.01); C07D 235/16 (2013.01); C07D 235/20 (2013.01); C07D 333/08 (2013.01); C07D 401/12 (2013.01); C07D 409/12 (2013.01)

Citation (search report)

See references of WO 9924407A1

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

DOCDB simple family (publication)

WO 9924407 A1 19990520; AU 1208999 A 19990531; EP 1030844 A1 20000830

DOCDB simple family (application)

US 9823362 W 19981103; AU 1208999 A 19981103; EP 98955238 A 19981103