Global Patent Index - EP 1030844 A1

EP 1030844 A1 2000-08-30 - COMPOUNDS WHICH INHIBIT TRYPTASE ACTIVITY

Title (en)

COMPOUNDS WHICH INHIBIT TRYPTASE ACTIVITY

Title (de)

VERBINDUNGEN, DIE DIE AKTIVITÄT VON TRYPTASE HEMMEN

Title (fr)

COMPOSES INHIBANT L'ACTIVITE DE LA TRYPTASE

Publication

EP 1030844 A1 (EN)

Application

EP 98955238 A

Priority

  • US 9823362 W
  • US 6515497 P
  • US 17969598 A

Abstract (en)

[origin: WO9924407A1] The present invention is directed to compounds which are capable of inhibiting the activity of tryptase. Such compounds are useful in the treatment or prevention of inflammatory disease, particularly those disease states which are mediated by mast cell activation. Also encompassed by the invention are formulations comprising the noted compounds, processes for preparing such compounds and methods for treating or preventing an inflammatory disease.

IPC 1-7 (main, further and additional classification)

C07D 235/16; A61K 31/155; A61K 31/38; A61K 31/40; A61K 31/415; C07C 257/18; C07D 209/08; C07D 209/18; C07D 209/42; C07D 235/14; C07D 333/60; C07D 333/62; C07D 401/12; C07D 403/12; C07D 409/12

IPC 8 full level (invention and additional information)

C07C 257/18 (2006.01); C07D 209/08 (2006.01); C07D 235/16 (2006.01); C07D 235/20 (2006.01); C07D 333/08 (2006.01); C07D 401/12 (2006.01); C07D 409/12 (2006.01)

CPC (invention and additional information)

C07D 401/12 (2013.01); C07C 257/18 (2013.01); C07D 209/08 (2013.01); C07D 235/16 (2013.01); C07D 235/20 (2013.01); C07D 333/08 (2013.01); C07D 409/12 (2013.01)

Citation (search report)

See references of WO 9924407A1

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

EPO simple patent family

WO 9924407 A1 19990520; AU 1208999 A 19990531; EP 1030844 A1 20000830

INPADOC legal status


2001-11-21 [18D] DEEMED TO BE WITHDRAWN

- Effective date: 20010503

2001-02-07 [17Q] FIRST EXAMINATION REPORT

- Effective date: 20001221

2000-08-30 [17P] REQUEST FOR EXAMINATION FILED

- Effective date: 20000608

2000-08-30 [AK] DESIGNATED CONTRACTING STATES:

- Kind Code of Ref Document: A1

- Designated State(s): AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

2000-08-30 [AX] REQUEST FOR EXTENSION OF THE EUROPEAN PATENT TO

- Free text: AL PAYMENT 20000608;LT PAYMENT 20000608;LV PAYMENT 20000608;MK PAYMENT 20000608;RO PAYMENT 20000608;SI PAYMENT 20000608