EP 1040095 B1 20030416 - CYCLOHEXENE CARBOXYLATES AS NEURAMINIDASE INHIBITORS
Title (en)
CYCLOHEXENE CARBOXYLATES AS NEURAMINIDASE INHIBITORS
Title (de)
CYCLOHEXENCARBOXYLATE ALS INHIBITOREN DER NEURAMINIDASE
Title (fr)
CARBOXYLATES DE CYCLOHEXENE UTILISES COMME INHIBITEURS DE NEURAMINIDASE
Publication
Application
Priority
- US 9826327 W 19981210
- US 6955397 P 19971212
Abstract (en)
[origin: WO9931047A1] Novel compounds of Formula (I) are described. R<1>, R<2>, R<3>, R<4>, R<5> and R<6> are described in this specification. Synthetic intermediates and pharmaceutical compositions comprising the inhibitors of the invention are also described. Methods of inhibiting neuraminidase in samples suspected of containing neuraminidase are also described. Assay methods for detecting neuraminidase activity are also described.
IPC 1-7
C07C 233/52; C07C 69/75; C07C 69/757; A61K 31/16; A61K 31/215
IPC 8 full level
C07D 295/14 (2006.01); A61K 31/195 (2006.01); A61K 31/215 (2006.01); A61K 31/5375 (2006.01); A61P 31/16 (2006.01); A61P 43/00 (2006.01); C07C 233/52 (2006.01); C07C 247/14 (2006.01); C07C 271/24 (2006.01); C07C 309/66 (2006.01); C07D 203/26 (2006.01); C07D 295/155 (2006.01); C07D 303/40 (2006.01); C07D 317/46 (2006.01)
CPC (source: EP US)
A61P 31/00 (2017.12 - EP); A61P 31/16 (2017.12 - EP); A61P 43/00 (2017.12 - EP); C07C 233/52 (2013.01 - EP US); C07C 247/14 (2013.01 - EP US); C07C 271/24 (2013.01 - EP US); C07D 203/26 (2013.01 - EP US); C07D 295/155 (2013.01 - EP US); C07D 303/40 (2013.01 - EP US); C07D 317/46 (2013.01 - EP US); C07B 2200/07 (2013.01 - EP US); C07C 2601/02 (2017.04 - EP US); C07C 2601/14 (2017.04 - EP US); C07C 2601/16 (2017.04 - EP US)
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
WO 9931047 A1 19990624; AR 015493 A1 20010502; AT E237582 T1 20030515; AU 1722699 A 19990705; CA 2313638 A1 19990624; CA 2313638 C 20080722; DE 69813616 D1 20030522; DE 69813616 T2 20040205; EP 1040095 A1 20001004; EP 1040095 B1 20030416; ES 2196636 T3 20031216; HK 1033932 A1 20011005; JP 2002508347 A 20020319; JP 4422895 B2 20100224; TW 477783 B 20020301; TW 480247 B 20020321; US 6111132 A 20000829; ZA 9811314 B 19990614
DOCDB simple family (application)
US 9826327 W 19981210; AR P980106313 A 19981211; AT 98962059 T 19981210; AU 1722699 A 19981210; CA 2313638 A 19981210; DE 69813616 T 19981210; EP 98962059 A 19981210; ES 98962059 T 19981210; HK 01102443 A 20010404; JP 2000538977 A 19981210; TW 87120362 A 19981208; TW 90111328 A 19981208; US 20864698 A 19981210; ZA 9811314 A 19981210