Global Patent Index - EP 1047689 A1

EP 1047689 A1 20001102 - SUBSTITUTED GUANIDINE DERIVATIVES AND THEIR USE FOR COMBATING ANIMAL PESTS

Title (en)

SUBSTITUTED GUANIDINE DERIVATIVES AND THEIR USE FOR COMBATING ANIMAL PESTS

Title (de)

SUBSTITUIERTE GUANIDIN-DERIVATE UND IHRE VERWENDUNG ZUR BEKÄMPFUNG VON TIERISCHEN SCHÄDLINGEN

Title (fr)

DERIVES DE GUANIDINE SUBSTITUES ET LEUR UTILISATION POUR LUTTER CONTRE LES PARASITES ANIMAUX

Publication

EP 1047689 A1 20001102 (DE)

Application

EP 98966405 A 19981224

Priority

  • DE 19800400 A 19980108
  • EP 9808444 W 19981224

Abstract (en)

[origin: DE19800400A1] The present invention relates to novel guanidine derivatives of formula (1), wherein R<1> represents a five or six membered heterocyclic group containing 1, 2, 3 or 4 nitrogen atoms and/or one or two oxygen or sulphur atoms as heteroatom ring members, whereby the number of heteroatoms is 1, 2, 3 or 4 and is optionally substituted by halogen, cyano, nitro, alkyl, halogen alkane, alkenyl, halogen alkenyl, alkinyl, alkoxy, halogen alkoxy, alkenyloxy, halogen alkenyloxy, alkinyloxy, alkylthio, halogen alkanethio, alkenylthio, halogen alkenylthio, alkinylthio, alkylsulphinyl, halogen alkanesulphinyl, alkylsulphonyl, amino, alkylamino, dialkylamino, aryl, arylthio, arylamino, aralkyl, formylamino, alkylcarbonylamino, formyl, carbamoyl, alkylcarbonyl and or alkoxycarbonyl, R<2> represents hydrogen or alkyl, R<3> represents groups -OCR<4>, -OCOR<5>, OCOOR<6>, OCONR<7>R<8> and -OSO<2>R<9>, whereby R<4> and R<6> represent independently of each other alkyl, alkoxyalkyl, halogen alkane, alkenyl, alkinyl, alkylaminoalkyl, dialkylaminoalkyl, optionally substituted cycloalkyl and optionally substituted phenyl or benzyl, R<7> and R<8> represent independently of each other hydrogen, alkyl, alkenyl and optionally substituted phenyl or benzyl and R<9> represents alkyl or optionally substituted pheyl, A represents groups -CH2CH2-, (CH2)3 and -CH=CH- and Z represents cyano or nitro, with the proviso that when Z represents NO2 and A represents -CH2CH2, the radical R<2> represents hydrogen and the compound of formula (1), wherein R<1> corresponds to formula (II), R<2> = H, R<3> = OCH3, A = -CH2CH2- and Z = NO2, is excluded.

IPC 1-7

C07D 401/06; C07D 417/06; A01N 43/78; A01N 43/50

IPC 8 full level

A01N 43/50 (2006.01); A01N 43/78 (2006.01); A01N 47/40 (2006.01); A01N 51/00 (2006.01); C07D 401/06 (2006.01); C07D 417/06 (2006.01)

CPC (source: EP KR US)

A01N 47/40 (2013.01 - EP KR US); A01N 51/00 (2013.01 - EP KR US); C07D 401/06 (2013.01 - EP KR US); C07D 417/06 (2013.01 - EP KR US)

Citation (search report)

See references of WO 9935141A1

Designated contracting state (EPC)

AT BE CH DE ES FR GB IT LI NL

DOCDB simple family (publication)

DE 19800400 A1 19990715; AU 2275999 A 19990726; BR 9813241 A 20010102; CN 1191247 C 20050302; CN 1285827 A 20010228; CN 1550498 A 20041201; CN 1810807 A 20060802; EP 1047689 A1 20001102; JP 2002500222 A 20020108; KR 20010033372 A 20010425; US 2003119828 A1 20030626; US 6503912 B1 20030107; US 6667310 B2 20031223; WO 9935141 A1 19990715

DOCDB simple family (application)

DE 19800400 A 19980108; AU 2275999 A 19981224; BR 9813241 A 19981224; CN 200410039993 A 19981224; CN 200510118649 A 19981224; CN 98812980 A 19981224; EP 9808444 W 19981224; EP 98966405 A 19981224; JP 2000527541 A 19981224; KR 20007006839 A 20000620; US 26185502 A 20021001; US 58267900 A 20000628