EP 1047698 A1 20001102 - PIPERAZINO DERIVATIVES AS NEUROKININ ANTAGONISTS
Title (en)
PIPERAZINO DERIVATIVES AS NEUROKININ ANTAGONISTS
Title (de)
PIPERAZINDERIVATE ALS NEUROKININ ANTAGONISTEN
Title (fr)
DERIVES DE LA PIPERAZINE EN TANT QU'ANTAGONISTES DE LA NEUROKININE
Publication
Application
Priority
- US 9900046 W 19990111
- US 694298 A 19980114
Abstract (en)
[origin: WO9936424A1] The invention relates to neurokinin antagonists of formula (I) wherein Z, Rc, y, m, u, Ar2, n, X, Rc', I and Ar2 are as described herein. These compounds are useful in the treatment of diseases such as asthma, anxiety, depression, emesis and nociception.
IPC 1-7
IPC 8 full level
A61K 31/496 (2006.01); A61P 11/00 (2006.01); A61P 11/06 (2006.01); A61P 11/14 (2006.01); A61P 17/00 (2006.01); A61P 17/04 (2006.01); A61P 17/06 (2006.01); A61P 25/00 (2006.01); A61P 25/16 (2006.01); A61P 25/22 (2006.01); A61P 29/00 (2006.01); A61P 43/00 (2006.01); C07D 471/08 (2006.01); C07D 487/08 (2006.01)
CPC (source: EP)
A61P 11/00 (2017.12); A61P 11/06 (2017.12); A61P 11/14 (2017.12); A61P 17/00 (2017.12); A61P 17/04 (2017.12); A61P 17/06 (2017.12); A61P 25/00 (2017.12); A61P 25/16 (2017.12); A61P 25/22 (2017.12); A61P 29/00 (2017.12); A61P 43/00 (2017.12); C07D 471/08 (2013.01); C07D 487/08 (2013.01); Y02P 20/582 (2015.11)
Citation (search report)
See references of WO 9936424A1
Designated contracting state (EPC)
AT BE CH DE DK ES FI FR GB GR IE IT LI LU NL PT SE
DOCDB simple family (publication)
WO 9936424 A1 19990722; AR 014950 A1 20010411; AU 2101399 A 19990802; CA 2317760 A1 19990722; CN 1135232 C 20040121; CN 1305481 A 20010725; CO 5080777 A1 20010925; EP 1047698 A1 20001102; JP 2002509151 A 20020326; PE 20000173 A1 20000309; ZA 99171 B 19990712
DOCDB simple family (application)
US 9900046 W 19990111; AR P990100086 A 19990111; AU 2101399 A 19990111; CA 2317760 A 19990111; CN 99802156 A 19990111; CO 99001260 A 19990112; EP 99901277 A 19990111; JP 2000540140 A 19990111; PE 00002199 A 19990111; ZA 99171 A 19990111