EP 1049472 A4 20020403 - ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE
Title (en)
ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE
Title (de)
ANTAGONISTEN DES GONADOTROPIN FREISETZENDEN HORMONS
Title (fr)
ANTAGONISTES DE LA GONADOLIBERINE
Publication
Application
Priority
- GB 9806694 A 19980327
- US 9822487 W 19981023
- US 6331297 P 19971028
Abstract (en)
[origin: WO9921557A1] There are disclosed compounds of formula (I) and pharmaceutically acceptable salts thereof which are useful as antagnoists of GnRH and as such may be useful for the treatment of a variety of sex-hormone related and other conditions in both men and women.
IPC 1-7
A61K 31/47; A61K 31/445; A61K 31/405; A61K 31/38; A61K 31/35; C07D 209/04; C07D 209/14; C07D 333/52; C07D 409/14; C07D 401/10; C07D 209/18; C07D 209/42; A61P 5/24
IPC 8 full level
C07D 217/12 (2006.01); A61K 31/403 (2006.01); A61K 31/404 (2006.01); A61K 31/405 (2006.01); A61K 31/4427 (2006.01); A61K 31/443 (2006.01); A61K 31/4433 (2006.01); A61K 31/454 (2006.01); A61K 31/472 (2006.01); A61K 31/4725 (2006.01); A61P 1/00 (2006.01); A61P 13/08 (2006.01); A61P 15/00 (2006.01); A61P 15/18 (2006.01); A61P 19/08 (2006.01); A61P 35/00 (2006.01); A61P 43/00 (2006.01); C07D 209/14 (2006.01); C07D 401/10 (2006.01); C07D 401/14 (2006.01); C07D 405/10 (2006.01); C07D 405/14 (2006.01); C07D 409/10 (2006.01); C07D 409/14 (2006.01)
CPC (source: EP)
A61P 1/00 (2017.12); A61P 5/24 (2017.12); A61P 13/08 (2017.12); A61P 15/00 (2017.12); A61P 15/18 (2017.12); A61P 19/08 (2017.12); A61P 35/00 (2017.12); A61P 43/00 (2017.12); C07D 209/14 (2013.01)
Citation (search report)
- [X] FR 2181559 A1 19731207 - AEC CHIMIE ORGANIQUE BIO [FR]
- [X] GB 1562825 A 19800319 - LILLY CO ELI
- [XD] WO 9721703 A1 19970619 - MERCK & CO INC [US], et al & WO 9721704 A1 19970619 - MERCK & CO INC [US], et al
- [XD] US 5030640 A 19910709 - FISHER MICHAEL H [US], et al
- [XD] US 4544663 A 19851001 - MANNING ROBERT E [US], et al
- [E] WO 9855119 A1 19981210 - MERCK & CO INC [US], et al
- See references of WO 9921557A1
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU NL PT SE
DOCDB simple family (publication)
WO 9921557 A1 19990506; AU 1197299 A 19990517; CA 2308069 A1 19990506; EP 1049472 A1 20001108; EP 1049472 A4 20020403; JP 2001520997 A 20011106
DOCDB simple family (application)
US 9822487 W 19981023; AU 1197299 A 19981023; CA 2308069 A 19981023; EP 98955082 A 19981023; JP 2000517715 A 19981023