Global Patent Index - EP 1052982 A4

EP 1052982 A4 20041006 - AMINOTETRALINS AS 5-HT 1D$g(a)? AGONISTS

Title (en)

AMINOTETRALINS AS 5-HT 1D$g(a)? AGONISTS

Title (de)

AMINOTETRALINE ALS 5HT1D-alpha AGONISTEN

Title (fr)

AMINOTETRALINES SERVANT D'AGONISTES DE 5-HT 1D$g(a)?

Publication

EP 1052982 A4 20041006 (EN)

Application

EP 98918773 A 19980427

Priority

  • US 9808436 W 19980427
  • US 84639997 A 19970430

Abstract (en)

[origin: WO9848786A1] A class of novel aminotetralins is disclosed useful as 5-HT1D alpha agonists.

[origin: WO9848786A1] A class of novel aminotetralins is disclosed useful as 5-HT1D alpha agonists.

IPC 1-7

A61K 31/135; A61K 31/335; A61K 31/34; A61K 31/35; C07C 211/42; C07D 305/08; C07D 305/10; C07D 307/22; C07D 307/30; C07D 309/14; C07D 309/28; C07D 313/04; C07D 313/18

IPC 8 full level

A61K 31/135 (2006.01); A61K 31/341 (2006.01); A61K 31/351 (2006.01); A61P 13/00 (2006.01); A61P 13/08 (2006.01); A61P 15/10 (2006.01); A61P 25/00 (2006.01); A61P 25/06 (2006.01); A61P 25/16 (2006.01); A61P 25/22 (2006.01); A61P 25/28 (2006.01); A61P 43/00 (2006.01); C07C 211/42 (2006.01); C07C 215/42 (2006.01); C07C 217/52 (2006.01); C07C 217/74 (2006.01); C07D 307/14 (2006.01); C07D 307/16 (2006.01); C07D 309/04 (2006.01)

CPC (source: EP)

A61K 31/135 (2013.01); A61K 31/341 (2013.01); A61K 31/351 (2013.01); A61P 13/00 (2017.12); A61P 13/08 (2017.12); A61P 15/10 (2017.12); A61P 25/00 (2017.12); A61P 25/06 (2017.12); A61P 25/16 (2017.12); A61P 25/22 (2017.12); A61P 25/28 (2017.12); A61P 43/00 (2017.12); C07C 211/42 (2013.01); C07C 215/42 (2013.01); C07C 217/74 (2013.01); C07D 307/14 (2013.01); C07D 309/04 (2013.01); C07C 2601/04 (2017.04); C07C 2601/08 (2017.04); C07C 2601/10 (2017.04); C07C 2601/16 (2017.04); C07C 2601/18 (2017.04); C07C 2602/10 (2017.04)

Citation (search report)

  • [Y] EP 0272534 A2 19880629 - BAYER AG [DE]
  • [Y] US 5571942 A 19961105 - HOECHSTETTER CRAIG S [US], et al
  • [Y] LIU Y. ET AL.: "C8-substituted derivatives of 2-(dipropylamino)tetralin: exploration of the effect of C8-aryl and heteroaryl substituents on the interaction with 5-HT1A-receptors", EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY., vol. 30, no. 4, 1995, FREDITIONS SCIENTIFIQUE ELSEVIER, PARIS., pages 277 - 286, XP002291176
  • See references of WO 9848786A1

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU NL PT SE

DOCDB simple family (publication)

WO 9848786 A1 19981105; AU 7163598 A 19981124; CA 2288897 A1 19981105; EP 1052982 A1 20001122; EP 1052982 A4 20041006; JP 2001524112 A 20011127

DOCDB simple family (application)

US 9808436 W 19980427; AU 7163598 A 19980427; CA 2288897 A 19980427; EP 98918773 A 19980427; JP 54724398 A 19980427