Global Patent Index - EP 1052992 A1

EP 1052992 A1 20001122 - CYCLIC AMINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY

Title (en)

CYCLIC AMINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY

Title (de)

CYCLISCHE AMINE MODULATOREN DER CHEMOKINREZEPTOREN

Title (fr)

AMINES CYCLIQUES UTILISEES EN TANT QUE MODULATEURS DE L'ACTIVITE DU RECEPTEUR DE CHEMOKINE

Publication

EP 1052992 A1 20001122 (EN)

Application

EP 99906697 A 19990201

Priority

  • GB 9810890 A 19980520
  • US 9902165 W 19990201
  • US 7344698 P 19980202

Abstract (en)

[origin: WO9938514A1] The present invention is directed to cyclic amines of formula I (wherein R<1>, R<2>, R<3>, m and n are defined herein) which are useful as modulators of chemokine receptor activity. In particular, these compounds are useful as modulators of the chemokine receptors CCR-1, CCR-2, CCR-2A, CCR-2B, CCR-3, CCR-4, CCR-5, CXCR-3, and/or CXCR-4.

IPC 1-7

A61K 31/445; A61K 31/535; A61K 31/54; A61K 31/55; C07D 211/18; C07D 211/32; C07D 211/36; C07D 211/96; C07D 401/06; C07D 401/14; C07D 407/14; C07D 409/10; C07D 409/14; C07D 413/14; C07D 417/14; C07D 471/10; C07D 491/107

IPC 8 full level

A61K 31/4427 (2006.01); A61K 31/443 (2006.01); A61K 31/4433 (2006.01); A61K 31/4468 (2006.01); A61K 31/4525 (2006.01); A61K 31/4535 (2006.01); A61K 31/454 (2006.01); A61P 31/18 (2006.01); A61P 37/04 (2006.01); A61P 43/00 (2006.01); C07D 211/56 (2006.01); C07D 211/58 (2006.01); C07D 401/06 (2006.01); C07D 405/06 (2006.01); C07D 405/12 (2006.01); C07D 409/06 (2006.01); C07D 409/12 (2006.01); C07D 491/107 (2006.01); C07D 521/00 (2006.01)

CPC (source: EP)

A61P 31/18 (2017.12); A61P 37/04 (2017.12); A61P 43/00 (2017.12); C07D 211/56 (2013.01); C07D 231/12 (2013.01); C07D 233/56 (2013.01); C07D 249/08 (2013.01); C07D 401/06 (2013.01); C07D 405/06 (2013.01); C07D 409/06 (2013.01)

Citation (search report)

See references of WO 9938514A1

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU NL PT SE

DOCDB simple family (publication)

WO 9938514 A1 19990805; AU 2654399 A 19990816; CA 2319781 A1 19990805; EP 1052992 A1 20001122; JP 2002501898 A 20020122

DOCDB simple family (application)

US 9902165 W 19990201; AU 2654399 A 19990201; CA 2319781 A 19990201; EP 99906697 A 19990201; JP 2000529247 A 19990201