EP 1056743 A1 20001206 - BENZAMINE DERIVATIVES
Title (en)
BENZAMINE DERIVATIVES
Title (de)
BENZAMIDINDERIVATE ALS KOAGULATIONSFAKTOR-XA-HEMMER
Title (fr)
DERIVES DE BENZAMIDINE UTILISES COMME INHIBITEURS DU FACTEUR DE COAGULATION Xa
Publication
Application
Priority
- DE 19755268 A 19971212
- EP 9807673 W 19981127
Abstract (en)
[origin: DE19755268A1] The invention relates to novel compounds of formula (1) wherein X, Y, W, R<1>, R<2>, R<3> and R<4> have the meaning cited in Claim 1. The inventive compounds are inhibitors of coagulation factor Xa and can be used in prophylaxis and/or therapy for thromboembolic diseases.
IPC 1-7
C07D 413/14; C07D 413/12; C07D 295/26; C07C 257/18; A61K 31/41; A61K 31/495; A61K 31/155
IPC 8 full level
A61K 31/155 (2006.01); A61K 31/18 (2006.01); A61K 31/195 (2006.01); A61K 31/422 (2006.01); A61K 31/4245 (2006.01); A61K 31/426 (2006.01); A61K 31/433 (2006.01); C07D 295/12 (2006.01); A61K 31/454 (2006.01); A61K 31/495 (2006.01); A61K 31/496 (2006.01); A61K 31/506 (2006.01); A61P 7/02 (2006.01); A61P 9/10 (2006.01); A61P 25/00 (2006.01); A61P 29/00 (2006.01); A61P 43/00 (2006.01); C07C 257/18 (2006.01); C07C 311/05 (2006.01); C07C 311/18 (2006.01); C07C 311/19 (2006.01); C07C 311/29 (2006.01); C07D 239/42 (2006.01); C07D 263/20 (2006.01); C07D 263/24 (2006.01); C07D 271/06 (2006.01); C07D 277/28 (2006.01); C07D 285/14 (2006.01); C07D 295/22 (2006.01); C07D 295/26 (2006.01); C07D 413/06 (2006.01); C07D 413/10 (2006.01); C07D 413/12 (2006.01); C07D 413/14 (2006.01); C07D 417/12 (2006.01); C07D 417/14 (2006.01)
CPC (source: EP KR)
A61P 7/02 (2018.01 - EP); A61P 9/10 (2018.01 - EP); A61P 25/00 (2018.01 - EP); A61P 29/00 (2018.01 - EP); A61P 43/00 (2018.01 - EP); C07C 257/18 (2013.01 - EP KR); C07C 311/05 (2013.01 - EP KR); C07C 311/18 (2013.01 - EP KR); C07D 263/16 (2013.01 - KR); C07D 263/20 (2013.01 - EP); C07D 295/26 (2013.01 - EP KR); C07D 413/10 (2013.01 - EP KR); C07D 417/14 (2013.01 - EP KR)
Designated contracting state (EPC)
AT BE CH DE DK ES FI FR GB GR IE IT LI LU NL PT SE
DOCDB simple family (publication)
WO 9931092 A1 19990624; AR 017844 A1 20011024; AU 1964799 A 19990705; AU 744002 B2 20020214; BR 9813477 A 20001024; CA 2313651 A1 19990624; CN 1281451 A 20010124; DE 19755268 A1 19990617; EP 1056743 A1 20001206; HU P0004353 A2 20020328; HU P0004353 A3 20020429; JP 2002508370 A 20020319; KR 20010032963 A 20010425; NO 20002958 D0 20000609; NO 20002958 L 20000811; PL 341008 A1 20010312; RU 2203897 C2 20030510; SK 8572000 A3 20010710; ZA 9811339 B 19990708
DOCDB simple family (application)
EP 9807673 W 19981127; AR P980106293 A 19981211; AU 1964799 A 19981127; BR 9813477 A 19981127; CA 2313651 A 19981127; CN 98812087 A 19981127; DE 19755268 A 19971212; EP 98964455 A 19981127; HU P0004353 A 19981127; JP 2000539016 A 19981127; KR 20007006310 A 20000609; NO 20002958 A 20000609; PL 34100898 A 19981127; RU 2000118792 A 19981127; SK 8572000 A 19981127; ZA 9811339 A 19981210