Global patent index - EP 1060164 A1

EP 1060164 A1 2000-12-20 - META-AZACYCLIC AMINO BENZOIC ACID COMPOUNDS AND DERIVATIVES THEREOF BEING INTEGRIN ANTAGONISTS

Title (en)

META-AZACYCLIC AMINO BENZOIC ACID COMPOUNDS AND DERIVATIVES THEREOF BEING INTEGRIN ANTAGONISTS

Title (de)

META-AZACYKLISCHE AMINO BENZOSÄURE DERIVATE MIT INTEGRIN ANTAGONISCHER WIRKUNG

Title (fr)

COMPOSES D'ACIDE META-AZACYCLIQUE AMINO BENZOIQUE ET DERIVES ANTAGONISTES DE L'INTEGRINE

Publication

EP 1060164 A1 (EN)

Application

EP 99937927 A

Priority

  • US 9903281 W
  • US 3427098 A

Abstract (en)

[origin: WO9944994A1] The present invention is directed to compounds of formula (1) and pharmaceutically acceptable salts and isomers thereof useful as alpha v beta 3 integrin antagonists.

IPC 1-7 (main, further and additional classification)

C07D 233/26; A61K 31/505

IPC 8 full level (invention and additional information)

A61K 31/505 (2006.01); A61K 31/675 (2006.01); A61K 31/70 (2006.01); A61P 3/14 (2006.01); A61P 9/00 (2006.01); A61P 19/02 (2006.01); A61P 19/08 (2006.01); A61P 29/00 (2006.01); A61P 35/00 (2006.01); A61P 35/04 (2006.01); A61P 43/00 (2006.01); C07D 239/14 (2006.01)

CPC (invention and additional information)

A61K 31/704 (2013.01); A61K 31/505 (2013.01); A61K 31/675 (2013.01); C07D 239/14 (2013.01)

Combination set (CPC)

  1. A61K 31/505 + A61K 2300/00
  2. A61K 31/675 + A61K 2300/00
  3. A61K 31/704 + A61K 2300/00

Citation (search report)

See references of WO 9944994A1

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

EPO simple patent family

WO 9944994 A1 19990910; AP 1244 A 20040204; AP 200001893 D0 20000930; AR 018139 A1 20011031; AU 3294799 A 19990920; AU 753230 B2 20021010; BG 104740 A 20010228; BR 9908470 A 20001205; CA 2322207 A1 19990910; CN 1214011 C 20050810; CN 1291978 A 20010418; EE 200000506 A 20020415; EP 1060164 A1 20001220; GE P20033118 B 20030610; HR P20000574 A2 20010831; HU 0100865 A2 20010828; HU 0100865 A3 20011128; ID 25591 A 20001019; IL 137653 D0 20011031; IS 5582 A 20000804; JP 2002505323 A 20020219; MY 123908 A 20060630; NO 20004316 A 20001106; NO 20004316 D0 20000830; NO 315703 B1 20031013; NZ 506598 A 20030725; OA 11530 A 20040517; PL 342726 A1 20010702; SK 13002000 A3 20010710; TR 200002542 T2 20010521; UA 71906 C2 20001115; YU 52000 A 20030228; ZA 9904406 B 20000211

INPADOC legal status

2009-03-04 [18D] DEEMED TO BE WITHDRAWN

- Ref Legal Event Code: 18D

- Effective date: 20080830

2008-11-26 [D18D] EP-APPLICATION DEEMED TO BE WITHDRAWN: (DELETED)

- Ref Legal Event Code: D18D

2003-07-09 [17Q] FIRST EXAMINATION REPORT

- Ref Legal Event Code: 17Q

- Effective date: 20030522

2000-12-20 [17P] REQUEST FOR EXAMINATION FILED

- Ref Legal Event Code: 17P

- Effective date: 20000929

2000-12-20 [AK] DESIGNATED CONTRACTING STATES:

- Ref Legal Event Code: AK

- Designated State(s): AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

2000-12-20 [AX] REQUEST FOR EXTENSION OF THE EUROPEAN PATENT TO

- Ref Legal Event Code: AX

- Free Format Text: AL PAYMENT 20000929;LT PAYMENT 20000929;LV PAYMENT 20000929;MK PAYMENT 20000929;RO PAYMENT 20000929;SI PAYMENT 20000929