Global Patent Index - EP 1062222 A1

EP 1062222 A1 20001227 - SERINE PEPTIDASE MODULATORS

Title (en)

SERINE PEPTIDASE MODULATORS

Title (de)

SERIN-PEPTIDASE MODULATOREN

Title (fr)

MODULATEURS DE LA SERINE PEPTIDASE

Publication

EP 1062222 A1 20001227 (EN)

Application

EP 99911781 A 19990309

Priority

  • EP 99911781 A 19990309
  • EP 9901617 W 19990309
  • EP 98200733 A 19980309

Abstract (en)

[origin: WO9946272A1] The present invention relates to new compounds having modulatory (inhibitory and stimulatory) activity on serine peptidases and proteases in general and dipeptidyl peptidase IV, prolyl oligopeptidase (PO), dipeptidyl peptidase II (DPP II), fibroblast activation protein alpha (FAP alpha ), lysosomal Pro-X carboxypeptidase and elastase in particular. These new compounds can be used for the treatment of a variety of disease states in which these peptidases are involved.

IPC 1-7

C07F 9/572; A61K 31/675; G01N 33/58; C07F 9/40; C07F 9/6571

IPC 8 full level

A61K 31/675 (2006.01); A61P 1/00 (2006.01); A61P 3/04 (2006.01); A61P 3/10 (2006.01); A61P 7/02 (2006.01); A61P 9/00 (2006.01); A61P 11/00 (2006.01); A61P 19/08 (2006.01); A61P 25/00 (2006.01); A61P 25/04 (2006.01); A61P 29/00 (2006.01); A61P 35/00 (2006.01); A61P 37/02 (2006.01); A61P 37/06 (2006.01); A61P 43/00 (2006.01); C07F 9/40 (2006.01); C07F 9/572 (2006.01); C07F 9/6571 (2006.01); G01N 33/58 (2006.01)

CPC (source: EP)

A61P 1/00 (2017.12); A61P 3/04 (2017.12); A61P 3/10 (2017.12); A61P 7/02 (2017.12); A61P 9/00 (2017.12); A61P 11/00 (2017.12); A61P 19/08 (2017.12); A61P 25/00 (2017.12); A61P 25/04 (2017.12); A61P 29/00 (2017.12); A61P 35/00 (2017.12); A61P 37/02 (2017.12); A61P 37/06 (2017.12); A61P 43/00 (2017.12); C07F 9/4006 (2013.01); C07F 9/572 (2013.01); C07F 9/657181 (2013.01)

Citation (search report)

See references of WO 9946272A1

Designated contracting state (EPC)

AT BE CH DE DK ES FI FR GB GR IE IT LI NL PT SE

DOCDB simple family (publication)

WO 9946272 A1 19990916; AU 3034299 A 19990927; EP 1062222 A1 20001227; JP 2002506075 A 20020226

DOCDB simple family (application)

EP 9901617 W 19990309; AU 3034299 A 19990309; EP 99911781 A 19990309; JP 2000535649 A 19990309