Global Patent Index - EP 1062222 A1

EP 1062222 A1 2000-12-27 - SERINE PEPTIDASE MODULATORS

Title (en)

SERINE PEPTIDASE MODULATORS

Title (de)

SERIN-PEPTIDASE MODULATOREN

Title (fr)

MODULATEURS DE LA SERINE PEPTIDASE

Publication

EP 1062222 A1 (EN)

Application

EP 99911781 A

Priority

  • EP 99911781 A
  • EP 9901617 W
  • EP 98200733 A

Abstract (en)

[origin: WO9946272A1] The present invention relates to new compounds having modulatory (inhibitory and stimulatory) activity on serine peptidases and proteases in general and dipeptidyl peptidase IV, prolyl oligopeptidase (PO), dipeptidyl peptidase II (DPP II), fibroblast activation protein alpha (FAP alpha ), lysosomal Pro-X carboxypeptidase and elastase in particular. These new compounds can be used for the treatment of a variety of disease states in which these peptidases are involved.

IPC 1-7 (main, further and additional classification)

C07F 9/572; A61K 31/675; C07F 9/40; C07F 9/6571; G01N 33/58

IPC 8 full level (invention and additional information)

A61K 31/675 (2006.01); A61P 1/00 (2006.01); A61P 3/04 (2006.01); A61P 3/10 (2006.01); A61P 7/02 (2006.01); A61P 9/00 (2006.01); A61P 11/00 (2006.01); A61P 19/08 (2006.01); A61P 25/00 (2006.01); A61P 25/04 (2006.01); A61P 29/00 (2006.01); A61P 35/00 (2006.01); A61P 37/02 (2006.01); A61P 37/06 (2006.01); A61P 43/00 (2006.01); C07F 9/40 (2006.01); C07F 9/572 (2006.01); C07F 9/6571 (2006.01); G01N 33/58 (2006.01)

CPC (invention and additional information)

C07F 9/657181 (2013.01); C07F 9/4006 (2013.01); C07F 9/5726 (2013.01)

Citation (search report)

See references of WO 9946272A1

Designated contracting state (EPC)

AT BE CH DE DK ES FI FR GB GR IE IT LI NL PT SE

EPO simple patent family

WO 9946272 A1 19990916; AU 3034299 A 19990927; EP 1062222 A1 20001227; JP 2002506075 A 20020226

INPADOC legal status


2003-12-03 [18D] DEEMED TO BE WITHDRAWN

- Effective date: 20030520

2001-08-22 [17Q] FIRST EXAMINATION REPORT

- Effective date: 20010704

2000-12-27 [17P] REQUEST FOR EXAMINATION FILED

- Effective date: 20000919

2000-12-27 [AK] DESIGNATED CONTRACTING STATES:

- Kind Code of Ref Document: A1

- Designated State(s): AT BE CH DE DK ES FI FR GB GR IE IT LI NL PT SE

2000-12-27 [AX] REQUEST FOR EXTENSION OF THE EUROPEAN PATENT TO

- Free text: LT PAYMENT 20000919;LV PAYMENT 20000919;SI PAYMENT 20000919