Global Patent Index - EP 1073624 A1

EP 1073624 A1 20010207 - AMINOMETHYL-BENZOIC ESTER DERIVATIVES AS TRYPTASE INHIBITORS

Title (en)

AMINOMETHYL-BENZOIC ESTER DERIVATIVES AS TRYPTASE INHIBITORS

Title (de)

AMINOMETHYLBENZOESÄUREESTERDERIVATE ALS TRYPTASE INHIBITORE

Title (fr)

DERIVES D'ESTER AMINOMETHYL BENZOIQUE UTILISES COMME INHIBITEURS DE LA TRYPTASE

Publication

EP 1073624 A1 20010207 (EN)

Application

EP 99918168 A 19990423

Priority

  • GB 9901263 W 19990423
  • GB 9808813 A 19980424
  • GB 9822432 A 19981014

Abstract (en)

[origin: WO9955661A1] The invention relates to the use of compounds of formula (I) wherein R represents hydrogen, alkyl, alkenyl, hydroxy, alkoxy, aminoalkyl, hydroxyalkyl, carboxyalkyl, alkoxyalkyl, amino, halo, cyano, nitro, thiol, alkylthio, haloalkoxy or haloalkyl; Ar represents an optionally substituted carbocyclic or heterocyclic aryl group with the proviso that when Ar represents a naphthyl moiety it is not substituted by amidino or guanidine; and Y represents a hydrogen atom or alkyl group; or a physiologically tolerable salt thereof; for use as tryptase inhibitors.

IPC 1-7

C07C 229/38; A61K 31/24

IPC 8 full level

A61K 31/24 (2006.01); A61K 31/277 (2006.01); A61K 31/445 (2006.01); A61K 31/47 (2006.01); C07C 229/38 (2006.01); C07C 233/47 (2006.01); C07C 235/52 (2006.01); C07C 235/74 (2006.01); C07C 235/78 (2006.01); C07C 255/55 (2006.01); C07C 311/29 (2006.01); C07C 311/51 (2006.01); C07D 207/16 (2006.01); C07D 211/62 (2006.01); C07D 213/65 (2006.01); C07D 215/32 (2006.01); C07D 217/02 (2006.01); C07D 257/04 (2006.01); C07D 295/185 (2006.01); C07D 295/192 (2006.01)

CPC (source: EP)

A61K 31/24 (2013.01); A61K 31/277 (2013.01); A61K 31/445 (2013.01); A61K 31/47 (2013.01); C07C 229/38 (2013.01); C07C 233/47 (2013.01); C07C 235/52 (2013.01); C07C 235/74 (2013.01); C07C 235/78 (2013.01); C07C 255/55 (2013.01); C07C 311/29 (2013.01); C07C 311/51 (2013.01); C07D 207/16 (2013.01); C07D 211/62 (2013.01); C07D 213/65 (2013.01); C07D 215/32 (2013.01); C07D 217/02 (2013.01); C07D 257/04 (2013.01); C07D 295/185 (2013.01); C07D 295/192 (2013.01)

Citation (search report)

See references of WO 9955661A1

Designated contracting state (EPC)

CH DE ES FR GB IT LI SE

DOCDB simple family (publication)

WO 9955661 A1 19991104; AU 3620099 A 19991116; EP 1073624 A1 20010207

DOCDB simple family (application)

GB 9901263 W 19990423; AU 3620099 A 19990423; EP 99918168 A 19990423