EP 1073624 A1 20010207 - AMINOMETHYL-BENZOIC ESTER DERIVATIVES AS TRYPTASE INHIBITORS
Title (en)
AMINOMETHYL-BENZOIC ESTER DERIVATIVES AS TRYPTASE INHIBITORS
Title (de)
AMINOMETHYLBENZOESÄUREESTERDERIVATE ALS TRYPTASE INHIBITORE
Title (fr)
DERIVES D'ESTER AMINOMETHYL BENZOIQUE UTILISES COMME INHIBITEURS DE LA TRYPTASE
Publication
Application
Priority
- GB 9901263 W 19990423
- GB 9808813 A 19980424
- GB 9822432 A 19981014
Abstract (en)
[origin: WO9955661A1] The invention relates to the use of compounds of formula (I) wherein R represents hydrogen, alkyl, alkenyl, hydroxy, alkoxy, aminoalkyl, hydroxyalkyl, carboxyalkyl, alkoxyalkyl, amino, halo, cyano, nitro, thiol, alkylthio, haloalkoxy or haloalkyl; Ar represents an optionally substituted carbocyclic or heterocyclic aryl group with the proviso that when Ar represents a naphthyl moiety it is not substituted by amidino or guanidine; and Y represents a hydrogen atom or alkyl group; or a physiologically tolerable salt thereof; for use as tryptase inhibitors.
IPC 1-7
IPC 8 full level
A61K 31/24 (2006.01); A61K 31/277 (2006.01); A61K 31/445 (2006.01); A61K 31/47 (2006.01); C07C 229/38 (2006.01); C07C 233/47 (2006.01); C07C 235/52 (2006.01); C07C 235/74 (2006.01); C07C 235/78 (2006.01); C07C 255/55 (2006.01); C07C 311/29 (2006.01); C07C 311/51 (2006.01); C07D 207/16 (2006.01); C07D 211/62 (2006.01); C07D 213/65 (2006.01); C07D 215/32 (2006.01); C07D 217/02 (2006.01); C07D 257/04 (2006.01); C07D 295/185 (2006.01); C07D 295/192 (2006.01)
CPC (source: EP)
A61K 31/24 (2013.01); A61K 31/277 (2013.01); A61K 31/445 (2013.01); A61K 31/47 (2013.01); C07C 229/38 (2013.01); C07C 233/47 (2013.01); C07C 235/52 (2013.01); C07C 235/74 (2013.01); C07C 235/78 (2013.01); C07C 255/55 (2013.01); C07C 311/29 (2013.01); C07C 311/51 (2013.01); C07D 207/16 (2013.01); C07D 211/62 (2013.01); C07D 213/65 (2013.01); C07D 215/32 (2013.01); C07D 217/02 (2013.01); C07D 257/04 (2013.01); C07D 295/185 (2013.01); C07D 295/192 (2013.01)
Citation (search report)
See references of WO 9955661A1
Designated contracting state (EPC)
CH DE ES FR GB IT LI SE
DOCDB simple family (publication)
WO 9955661 A1 19991104; AU 3620099 A 19991116; EP 1073624 A1 20010207
DOCDB simple family (application)
GB 9901263 W 19990423; AU 3620099 A 19990423; EP 99918168 A 19990423