Global patent index - EP 1076641 A1

EP 1076641 A1 2001-02-21 - INHIBITORS OF IMPDH ENZYME

Title (en)

INHIBITORS OF IMPDH ENZYME

Title (de)

IMPDH ENZYMINHIBITOREN

Title (fr)

INHIBITEURS DE L'ENZYME IMPDH

Publication

EP 1076641 A1 (EN)

Application

EP 99918831 A

Priority

  • US 9909005 W
  • US 8338598 P

Abstract (en)

[origin: WO9955663A1] The present invention relates to compounds which inhibit IMPDH. This invention also relates to pharmaceutical compositions comprising these compounds. The compounds and pharmaceutical compositions of this invention are particularly well suited for inhibiting IMPDH enzyme activity and consequently, may be advantageously used as therapeutic agents for IMPDH mediated processes. This invention also relates to methods for inhibiting the activity of IMPDH using the compounds of this invention and related compounds.

IPC 1-7 (main, further and additional classification)

C07C 235/56; A61K 31/135; A61K 31/165; A61K 31/18; A61K 31/395; C07C 217/84; C07C 311/21; C07D 263/32

IPC 8 full level (invention and additional information)

A61K 31/167 (2006.01); A61K 31/18 (2006.01); A61K 31/235 (2006.01); A61K 31/277 (2006.01); A61K 31/357 (2006.01); A61K 31/36 (2006.01); A61K 31/421 (2006.01); A61K 31/422 (2006.01); A61P 1/18 (2006.01); A61P 9/08 (2006.01); A61P 9/10 (2006.01); A61P 11/00 (2006.01); A61P 11/06 (2006.01); A61P 19/02 (2006.01); A61P 29/00 (2006.01); A61P 31/12 (2006.01); A61P 35/00 (2006.01); A61P 35/02 (2006.01); A61P 37/06 (2006.01); A61P 43/00 (2006.01); C07C 217/84 (2006.01); C07C 233/75 (2006.01); C07C 235/66 (2006.01); C07C 235/88 (2006.01); C07C 237/48 (2006.01); C07C 255/60 (2006.01); C07C 309/75 (2006.01); C07C 311/21 (2006.01); C07C 311/29 (2006.01); C07C 317/40 (2006.01); C07C 323/42 (2006.01); C07C 333/08 (2006.01); C07D 213/75 (2006.01); C07D 263/32 (2006.01); C07D 271/06 (2006.01); C07D 307/91 (2006.01); C07D 317/68 (2006.01); C07D 413/12 (2006.01)

CPC (invention and additional information)

C07D 213/75 (2013.01); A61K 31/167 (2013.01); A61K 31/18 (2013.01); C07C 217/84 (2013.01); C07C 233/75 (2013.01); C07C 235/66 (2013.01); C07C 235/88 (2013.01); C07C 237/48 (2013.01); C07C 255/60 (2013.01); C07C 311/21 (2013.01); C07D 263/32 (2013.01); C07D 271/06 (2013.01); C07D 307/91 (2013.01); C07D 317/68 (2013.01); C07D 413/12 (2013.01)

Citation (search report)

See references of WO 9955663A1

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

EPO simple patent family

WO 9955663 A1 19991104; AU 3665199 A 19991116; EP 1076641 A1 20010221; JP 2002512997 A 20020508

INPADOC legal status

2011-12-09 [REG HK WD] APPLICATIONS WITHDRAWN, DEEMED TO BE WITHDRAWN, OR REFUSED AFTER PUBLICATION IN HONG KONG

- Ref Legal Event Code: WD

- Ref Document Number: 1034955

- Country of Ref Document: HK

2011-04-27 [18D] DEEMED TO BE WITHDRAWN

- Ref Legal Event Code: 18D

- Effective date: 20101103

2002-11-06 [17Q] FIRST EXAMINATION REPORT

- Ref Legal Event Code: 17Q

- Effective date: 20020919

2001-02-21 [17P] REQUEST FOR EXAMINATION FILED

- Ref Legal Event Code: 17P

- Effective date: 20001128

2001-02-21 [AK] DESIGNATED CONTRACTING STATES:

- Ref Legal Event Code: AK

- Designated State(s): AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE