EP 1079763 A2 20010307 - SEROTONERGIC 5HT 7? RECEPTOR COMPOUNDS FOR TREATING OCULAR AND CNS DISORDERS
Title (en)
SEROTONERGIC 5HT 7? RECEPTOR COMPOUNDS FOR TREATING OCULAR AND CNS DISORDERS
Title (de)
VERBINDUNGEN DIE AUF DEN SEROTONERGISCHEN 5-HT7 REZEPTOR WIRKEN ZUR BEHANDLUNG VON SEHSTÖRUNGEN UND STÖRUNGEN DES CNS
Title (fr)
COMPOSES A AFFINITE POUR LE RECEPTEUR DE 5HT 7? SEROTONINERGIQUE, DESTINES AU TRAITEMENT DE TROUBLES OCULAIRES ET DU SYSTEME NERVEUX CENTRAL
Publication
Application
Priority
- US 9910179 W 19990510
- US 8600698 P 19980519
- US 8600598 P 19980519
- US 8598998 P 19980519
- US 8600298 P 19980519
Abstract (en)
[origin: WO9959499A2] Compounds with 5HT7 receptor affinity (some of which are novel) useful for lowering IOP, improving blood flow to the optic nerve head and the retina, providing neuroprotection, and treating retinal diseases are disclosed. The Compounds are also useful for treating sleep disorders, depression, and other psychiatric disorders, such as, schizophrenia, anxiety, obsessive compulsive disorder, circadian rhythm disorders, and centrally and peripherally mediated hypertension. Compositions and methods for their use are also disclosed.
IPC 1-7
IPC 8 full level
C07D 295/12 (2006.01); A61K 31/4427 (2006.01); A61K 31/4439 (2006.01); A61K 31/445 (2006.01); A61K 31/472 (2006.01); A61K 31/4725 (2006.01); A61K 31/495 (2006.01); A61K 31/496 (2006.01); A61K 31/542 (2006.01); A61P 9/12 (2006.01); A61P 25/18 (2006.01); A61P 25/20 (2006.01); A61P 25/22 (2006.01); A61P 25/24 (2006.01); A61P 27/02 (2006.01); A61P 43/00 (2006.01); C07D 209/08 (2006.01); C07D 211/22 (2006.01); C07D 217/04 (2006.01); C07D 295/088 (2006.01); C07D 295/13 (2006.01); C07D 401/12 (2006.01); C07D 513/04 (2006.01)
CPC (source: EP)
A61P 9/12 (2017.12); A61P 25/18 (2017.12); A61P 25/20 (2017.12); A61P 25/22 (2017.12); A61P 25/24 (2017.12); A61P 27/02 (2017.12); A61P 43/00 (2017.12); C07D 209/08 (2013.01); C07D 295/088 (2013.01); C07D 295/13 (2013.01); C07D 513/04 (2013.01)
Citation (search report)
See references of WO 9959499A2
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
WO 9959499 A2 19991125; WO 9959499 A3 20000316; AU 3978899 A 19991206; BR 9910590 A 20010123; CA 2332505 A1 19991125; CN 1301161 A 20010627; EP 1079763 A2 20010307; JP 2002515408 A 20020528
DOCDB simple family (application)
US 9910179 W 19990510; AU 3978899 A 19990510; BR 9910590 A 19990510; CA 2332505 A 19990510; CN 99806330 A 19990510; EP 99922894 A 19990510; JP 2000549166 A 19990510