Global Patent Index - EP 1083897 A1

EP 1083897 A1 2001-03-21 - HIV INTEGRASE INHIBITORS

Title (en)

HIV INTEGRASE INHIBITORS

Title (de)

HIV INTEGRASE-INHIBITOREN

Title (fr)

INHIBITEURS DE VIH INTEGRASE

Publication

EP 1083897 A1 (EN)

Application

EP 99926096 A

Priority

  • GB 9814930 A
  • US 9912095 W
  • US 8784598 P

Abstract (en)

[origin: WO9962513A1] Nitrogen-containing heteroaryl dioxo-butyric acid derivatives are described as inhibitors of HIV integrase and inhibitors of HIV replication. These compounds are useful in the prevention or treatment of infection by HIV and the treatment of AIDS, either as compounds, pharmaceutically acceptable salts, pharmaceutical composition ingredients, whether or not in combination with other antivirals, immunomodulators, antibiotics or vaccines. Methods of treating AIDS and methods of preventing or treating infection by HIV are also described.

IPC 1-7 (main, further and additional classification)

A61K 31/40; A61K 31/415; A61K 31/445; C07D 207/30; C07D 207/333; C07D 209/04; C07D 209/12; C07D 211/18; C07D 211/26; C07D 211/28; C07D 211/32; C07D 211/40; C07D 231/10; C07D 231/12; C07D 233/54; C07D 233/64; C07D 401/04

IPC 8 full level (invention and additional information)

A61K 31/40 (2006.01); A61K 31/403 (2006.01); A61K 31/404 (2006.01); A61K 31/415 (2006.01); A61K 31/4427 (2006.01); A61K 31/454 (2006.01); A61K 45/06 (2006.01); C07D 207/30 (2006.01); C07D 207/333 (2006.01); C07D 207/34 (2006.01); C07D 209/12 (2006.01); C07D 209/18 (2006.01); C07D 231/12 (2006.01); C07D 233/54 (2006.01); C07D 233/64 (2006.01); C07D 401/04 (2006.01); C07D 207/32 (2006.01)

CPC (invention and additional information)

C07D 207/333 (2013.01); A61K 31/40 (2013.01); A61K 45/06 (2013.01); C07D 207/34 (2013.01); C07D 209/12 (2013.01); C07D 231/12 (2013.01); C07D 401/04 (2013.01)

Combination set (CPC)

A61K 31/40 + A61K 2300/00

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU NL PT SE

EPO simple patent family

WO 9962513 A1 19991209; AU 4225699 A 19991220; AU 756826 B2 20030123; AU 756826 C 20030821; CA 2329134 A1 19991209; EP 1083897 A1 20010321; EP 1083897 A4 20030102; JP 2002516858 A 20020611

INPADOC legal status


2004-03-10 [18W] WITHDRAWN

- Effective date: 20040102

2003-01-02 [A4] SUPPLEMENTARY SEARCH REPORT

- Effective date: 20021115

2003-01-02 [AK] DESIGNATED CONTRACTING STATES:

- Kind Code of Ref Document: A4

- Designated State(s): AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU NL PT SE

2001-03-21 [17P] REQUEST FOR EXAMINATION FILED

- Effective date: 20010103

2001-03-21 [AK] DESIGNATED CONTRACTING STATES:

- Kind Code of Ref Document: A1

- Designated State(s): AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU NL PT SE

2001-03-21 [AX] REQUEST FOR EXTENSION OF THE EUROPEAN PATENT TO

- Free text: AL PAYMENT 20010103;LT PAYMENT 20010103;LV PAYMENT 20010103;MK PAYMENT 20010103;RO PAYMENT 20010103;SI PAYMENT 20010103