Global Patent Index - EP 1084130 A1

EP 1084130 A1 2001-03-21 - SUBSTITUTED FIVE MEMBERED HETEROCYCLIC COMPOUNDS, FUNGICIDAL COMPOSITIONS CONTAINING THEM AND METHODS OF MANUFACTURE THEREOF

Title (en)

SUBSTITUTED FIVE MEMBERED HETEROCYCLIC COMPOUNDS, FUNGICIDAL COMPOSITIONS CONTAINING THEM AND METHODS OF MANUFACTURE THEREOF

Title (de)

SUBSTITUTIERTE FÜNFGLIEDRIGE HETEROCYCLISCHE VERBINDUNGEN, DIESE ENTHALTENDE FUNGIZIDE ZUBEREITUNGEN UND VERFAHREN ZUR HERSTELLUNG DAVON

Title (fr)

COMPOSES HETEROCYCLIQUES SUBSTITUES A CINQ ELEMENTS, COMPOSITIONS FONGICIDES ET LEURS PROCEDES DE FABRICATION

Publication

EP 1084130 A1 (EN)

Application

EP 99927224 A

Priority

  • US 9912502 W
  • US 8839898 P

Abstract (en)

[origin: WO9962915A1] The fungicidal compound 4,5-dimethyl-N-2-propenyl-2-(trimethylsilyl)-3-thiophenecarboxamide (Formula (I)) has shown superior and unexpected control of the growth of the soil-borne fungus Gaeumannomyces graminis (Gg). The present invention provides a novel compound for synthesizing the compound of Formula (I) which uses the compound 4-hydroxy-4,5-dimethyl-2-trimethylsilanyl-dihydrothiophene-3-carboxylic acid allylamide (Formula (II)) as well as novel compounds of synthesizing the allylamide. In addition, Formula (II) itself has unexpectedly been found to provide control of Gg. Therefore, the compounds having Formula (III) or an agronomic salts and compositions thereof are expected to provide such control as well; wherein Q is -NH, S, or O; W is O, or S; X is -OH, -OAc, -OR, where R is lower alkyl; Y is S, O, or -NH; Z is -Si(R)3, -C(R)3, where R is lower alkyl; R1 is a lower alkyl, allyl, or propargyl; R2 is a lower alkyl or aryl; and R3 and R4 are independently chosen from hydrogen, a lower alkyl and aryl; optionally, R2 and R3 together form a 5- or 6-membered ring.

IPC 1-7 (main, further and additional classification)

C07F 7/08; A01N 43/10; A01N 55/00; C07D 333/38

IPC 8 full level (invention and additional information)

A01N 43/10 (2006.01); A01N 55/00 (2006.01); A01N 55/10 (2006.01); A01P 3/00 (2006.01); C07D 333/38 (2006.01); C07F 7/08 (2006.01)

CPC (invention and additional information)

C07F 7/083 (2013.01); C07D 333/38 (2013.01); C07F 7/0814 (2013.01)

Citation (search report)

See references of WO 9962915A1

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

EPO simple patent family

WO 9962915 A1 19991209; AT 223422 T 20020915; AU 4418399 A 19991220; AU 762985 B2 20030710; BR 9911624 A 20011030; BR 9911624 B1 20100713; CA 2334221 A1 19991209; CA 2334221 C 20081223; CN 100503594 C 20090624; CN 1182142 C 20041229; CN 1314907 A 20010926; CN 1623995 A 20050608; CZ 20004529 A3 20010613; CZ 299799 B6 20081126; DE 69902782 D1 20021010; DE 69902782 T2 20030528; DK 1084130 T3 20021021; EP 1084130 A1 20010321; EP 1084130 B1 20020904; ES 2183568 T3 20030316; PL 199097 B1 20080829; PL 345161 A1 20011203; PT 1084130 E 20030131; RU 2220973 C2 20040110; US 6140511 A 20001031; US 6291513 B1 20010918

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