Global Patent Index - EP 1086064 A2

EP 1086064 A2 2001-03-28 - DIRECTED COMBINATORIAL COMPOUND LIBRARY AND HIGH THROUGHPUT ASSAYS FOR SCREENING SAME

Title (en)

DIRECTED COMBINATORIAL COMPOUND LIBRARY AND HIGH THROUGHPUT ASSAYS FOR SCREENING SAME

Title (de)

GERICHTETE KOMBINATORISCHE VERBINDUNGSBIBLIOTHEK UND HOCHDURCHSATZ ASSAYS FÜR DEREN SCREENING

Title (fr)

BANQUE COMBINATOIRE ET DIRIGEE DE COMPOSES ET DOSAGES HAUT RENDEMENT PERMETTANT LEUR CRIBLAGE

Publication

EP 1086064 A2 (EN)

Application

EP 99927613 A

Priority

  • CA 9900550 W
  • US 8882898 P
  • US 12056299 P

Abstract (en)

[origin: WO9964378A2] A combinatorial library comprising a predetermined collection of nucleoside peptide molecules for inhibiting the transfer of a sugar from a selected sugar nucleotide donor to a selected acceptor by a carbohydrate processing enzyme. The nucleoside peptide molecule comprises (a) a nucleoside monomer; (b) a spacer monomer coupled to the nucleoside monomer wherein the spacer monomer comprises one or more amide linked amino acid residues, or a peptidomimetic; and (c) cap monomers attached to the spacer monomer. The nucleoside peptide molecules differ from each other as to the identity of at least one element of the nucleoside monomer, spacer monomer, or cap monomer.

IPC 1-7 (main, further and additional classification)

C07B 61/00; A61K 38/14; C07H 19/06; C07H 19/16; C07K 9/00; C12Q 1/48

IPC 8 full level (invention and additional information)

A61K 38/00 (2006.01); A61K 45/00 (2006.01); C07B 61/00 (2006.01); C07H 19/06 (2006.01); C07H 19/16 (2006.01); C07K 9/00 (2006.01); C12Q 1/48 (2006.01)

CPC (invention and additional information)

C07H 19/06 (2013.01); C07K 9/003 (2013.01); C12Q 1/48 (2013.01); C40B 40/00 (2013.01)

Citation (search report)

See references of WO 9964378A3

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

EPO simple patent family

WO 9964378 A2 19991216; WO 9964378 A3 20000921; AU 4493099 A 19991230; CA 2334338 A1 19991216; CN 1314913 A 20010926; EP 1086064 A2 20010328; JP 2002517474 A 20020618; MX PA00012237 A 20021115; NO 20006244 A 20010208; NO 20006244 D0 20001208

INPADOC legal status


2007-06-20 [18D] DEEMED TO BE WITHDRAWN

- Effective date: 20070103

2004-01-21 [RAP1] TRANSFER OF RIGHTS OF AN EP PUBLISHED APPLICATION

- Owner name: GLYCODESIGN HOLDINGS LTD.

2001-03-28 [17P] REQUEST FOR EXAMINATION FILED

- Effective date: 20001218

2001-03-28 [AK] DESIGNATED CONTRACTING STATES:

- Kind Code of Ref Document: A2

- Designated State(s): AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE