Global Patent Index - EP 1086091 A1

EP 1086091 A1 20010328 - HIV INTEGRASE INHIBITORS

Title (en)

HIV INTEGRASE INHIBITORS

Title (de)

HIV-INTEGRASE-INHIBITOREN

Title (fr)

INHIBITEURS DE VIH INTEGRASE

Publication

EP 1086091 A1 20010328 (EN)

Application

EP 99926095 A 19990601

Priority

  • GB 9814925 A 19980709
  • US 9912094 W 19990601
  • US 8784698 P 19980603

Abstract (en)

[origin: WO9962897A1] Sulfur-containing heteroaryl dioxo-butyric acid derivatives are described as inhibitors of HIV integrase and inhibitors of HIV replication. These compounds are useful in the prevention or treatment of infection by HIV and the treatment of AIDS, either as compounds, pharmaceutically acceptable salts, pharmaceutical composition ingredients, whether or not in combination with other antivirals, immunomodulators, antibiotics or vaccines. Methods of treating AIDS and methods of preventing or treating infection by HIV are also described.

IPC 1-7

C07D 333/74; C07D 333/56; C07D 333/22; C07D 277/04; C07D 277/18; A61K 31/38; A61K 31/425

IPC 8 full level

A61K 31/381 (2006.01); A61K 31/426 (2006.01); A61K 31/4433 (2006.01); A61K 31/4436 (2006.01); A61K 31/4535 (2006.01); A61P 31/18 (2006.01); A61P 37/04 (2006.01); A61P 43/00 (2006.01); C07D 277/20 (2006.01); C07D 277/34 (2006.01); C07D 277/36 (2006.01); C07D 277/38 (2006.01); C07D 277/42 (2006.01); C07D 333/24 (2006.01); C07D 333/28 (2006.01); C07D 333/32 (2006.01); C07D 333/34 (2006.01); C07D 333/36 (2006.01); C07D 333/56 (2006.01); C07D 333/60 (2006.01); C07D 333/74 (2006.01); C07D 409/12 (2006.01)

CPC (source: EP)

A61P 31/18 (2017.12); A61P 37/04 (2017.12); A61P 43/00 (2017.12); C07D 277/42 (2013.01); C07D 333/24 (2013.01); C07D 333/32 (2013.01); C07D 333/34 (2013.01); C07D 333/36 (2013.01); C07D 333/60 (2013.01); C07D 333/74 (2013.01); C07D 409/12 (2013.01)

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU NL PT SE

DOCDB simple family (publication)

WO 9962897 A1 19991209; AU 4225599 A 19991220; AU 757409 B2 20030220; CA 2333771 A1 19991209; EP 1086091 A1 20010328; EP 1086091 A4 20011010; JP 2002517390 A 20020618

DOCDB simple family (application)

US 9912094 W 19990601; AU 4225599 A 19990601; CA 2333771 A 19990601; EP 99926095 A 19990601; JP 2000552109 A 19990601