Global Patent Index - EP 1087938 A1

EP 1087938 A1 20010404 - INHIBITORS OF NEURAMINIDASES

Title (en)

INHIBITORS OF NEURAMINIDASES

Title (de)

NEURAMINIDASE INHIBITORE

Title (fr)

INHIBITEURS DE NEURAMINIDASES

Publication

EP 1087938 A1 20010404 (EN)

Application

EP 99918495 A 19990412

Priority

  • US 9907949 W 19990412
  • US 6580398 A 19980423

Abstract (en)

[origin: WO9954290A1] Disclosed are compounds of formula (I), (II) or (III), which are useful for inhibiting neuraminidases from disease-causing microorganisms, especially, influenza neuraminidase. Also disclosed are compositions and methods for preventing and treating diseases caused by microorganisms having a neuraminidase, processes for preparing the compounds and synthetic intermediates used in these processes.

IPC 1-7

C07C 271/24; C07C 233/52; C07C 233/47; C07C 271/22; C07D 233/54; C07D 263/32; A61K 31/33; A61K 31/16; C07C 237/24; C07D 307/24; C07D 405/04

IPC 8 full level

A61K 31/196 (2006.01); A61K 31/215 (2006.01); A61K 31/341 (2006.01); A61K 31/4164 (2006.01); A61K 31/421 (2006.01); A61P 31/16 (2006.01); A61P 43/00 (2006.01); C07C 233/47 (2006.01); C07C 233/52 (2006.01); C07C 237/24 (2006.01); C07C 271/22 (2006.01); C07C 271/24 (2006.01); C07D 233/54 (2006.01); C07D 263/32 (2006.01); C07D 307/24 (2006.01); C07D 317/32 (2006.01); C07D 405/04 (2006.01); C07D 493/08 (2006.01)

CPC (source: EP)

A61P 31/16 (2017.12); A61P 43/00 (2017.12); C07C 233/52 (2013.01); C07C 237/24 (2013.01); C07C 271/24 (2013.01); C07D 233/64 (2013.01); C07D 307/24 (2013.01); C07D 317/32 (2013.01); C07D 493/08 (2013.01); C07C 2601/08 (2017.04)

Citation (search report)

See references of WO 9954290A1

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU NL PT SE

DOCDB simple family (publication)

WO 9954290 A1 19991028; CA 2329660 A1 19991028; EP 1087938 A1 20010404; JP 2002521312 A 20020716

DOCDB simple family (application)

US 9907949 W 19990412; CA 2329660 A 19990412; EP 99918495 A 19990412; JP 2000544631 A 19990412