Global Patent Index - EP 1087950 A1

EP 1087950 A1 20010404 - NEW 2-AMINOCARBONYL-5(2H)-ISOXAZOLONES AS LIGANDS OF A DFP-BINDING SITE FOR TREATMENT OF CNS-DISEASES

Title (en)

NEW 2-AMINOCARBONYL-5(2H)-ISOXAZOLONES AS LIGANDS OF A DFP-BINDING SITE FOR TREATMENT OF CNS-DISEASES

Title (de)

NEUE 2-AMINOCARBONYL-5(2H)-ISOXAZOLONE ALS LIGANDEN EINER DFP-BINDUNGSSTELLE ZUR BEHANDLUNG VON ZNS-KRANKHEITEN

Title (fr)

NOUVELLES 2-AMINOCARBONYL-5(2H)-ISOXAZOLONES EN TANT QUE LIGANDS D'UN SITE DE LIAISON DE DFP POUR LE TRAITEMENT DE MALADIES DU SYSTEME NERVEUX CENTRAL

Publication

EP 1087950 A1 20010404 (DE)

Application

EP 99929179 A 19990611

Priority

  • DE 19827387 A 19980619
  • EP 9904030 W 19990611

Abstract (en)

[origin: DE19827387A1] The use of ligands of the high affinity binding site of diisopropyl-fluorophosphate (DFP) at mammalian brain membranes in the preparation of medicaments for prevention and treatment of central nervous system disorders, is new.

IPC 1-7

C07D 261/12; C07D 413/06; A61K 31/42

IPC 8 full level

A61K 31/42 (2006.01); A61K 31/422 (2006.01); A61K 31/423 (2006.01); A61K 31/454 (2006.01); A61K 31/496 (2006.01); A61K 31/5377 (2006.01); A61K 31/541 (2006.01); A61K 31/55 (2006.01); A61P 25/00 (2006.01); A61P 25/18 (2006.01); A61P 25/22 (2006.01); A61P 25/24 (2006.01); A61P 25/28 (2006.01); A61P 43/00 (2006.01); C07D 261/12 (2006.01); C07D 413/06 (2006.01)

CPC (source: EP US)

A61P 25/00 (2017.12 - EP); A61P 25/18 (2017.12 - EP); A61P 25/22 (2017.12 - EP); A61P 25/24 (2017.12 - EP); A61P 25/28 (2017.12 - EP); A61P 43/00 (2017.12 - EP); C07D 261/12 (2013.01 - EP US); C07D 413/06 (2013.01 - EP US)

Citation (search report)

See references of WO 9967229A1

Designated contracting state (EPC)

DE ES FR GB IT

DOCDB simple family (publication)

DE 19827387 A1 19991223; AU 4607999 A 20000110; CA 2335190 A1 19991229; EP 1087950 A1 20010404; JP 2002518490 A 20020625; US 6344471 B1 20020205; WO 9967229 A1 19991229

DOCDB simple family (application)

DE 19827387 A 19980619; AU 4607999 A 19990611; CA 2335190 A 19990611; EP 9904030 W 19990611; EP 99929179 A 19990611; JP 2000555883 A 19990611; US 72002401 A 20010227