Global patent index - EP 1087964 A1

EP 1087964 A1 2001-04-04 - N-BENZODIOXANYLMETHYL-1-PIPERIDYL-METHYLAMINE COMPOUNDS HAVING AFFINITY FOR 5-HT RECEPTORS

Title (en)

N-BENZODIOXANYLMETHYL-1-PIPERIDYL-METHYLAMINE COMPOUNDS HAVING AFFINITY FOR 5-HT RECEPTORS

Title (de)

N-BENZODIOXANYLMETHYL-1-PIPERIDYL-METHYLAMINVERBINDUNGEN MIT 5-HT-REZEPTORAFFINITÄT

Title (fr)

COMPOSES DE N-BENZODIOXANYLMETHYL-1-PIPERIDYL-METHYLAMINE PRESENTANT UNE AFFINITE POUR DES RECEPTEURS 5-HT

Publication

EP 1087964 A1 (EN)

Application

EP 99926434 A

Priority

  • EP 9903648 W
  • GB 9811879 A

Abstract (en)

[origin: WO9962902A1] Compounds of formula (I) including pharmaceutically acceptable salts thereof in which R represents H or F, their preparation and their use in the treatment of depression, anxiety, psychoses, Parkinson's disease, obesity, hypertension, Tourette's syndrome, sexual dysfunction, drug addiction, drug abuse, cognitive disorders, Alzheimer's disease, senile dementia, obsessive-compulsive behaviour, panic attacks, eating disorders, anorexia, cardiovascular and cerebrovascular disorders, migraine, non-insulin dependent diabetes melitus, hyperglycaemia, constipation, arrhythmia, disorders of the neuroendocrine system, stress, prostatic hypertrophy, drug-induced extrapyramidal symptoms or spasticity are described.

IPC 1-7 (main, further and additional classification)

C07D 405/12; A61K 31/335; C07D 319/20

IPC 8 full level (invention and additional information)

C07D 319/20 (2006.01); A61K 31/443 (2006.01); A61K 31/453 (2006.01); A61P 3/04 (2006.01); A61P 3/10 (2006.01); A61P 9/00 (2006.01); A61P 9/06 (2006.01); A61P 9/12 (2006.01); A61P 13/08 (2006.01); A61P 15/00 (2006.01); A61P 25/00 (2006.01); A61P 25/06 (2006.01); A61P 25/08 (2006.01); A61P 25/16 (2006.01); A61P 25/18 (2006.01); A61P 25/22 (2006.01); A61P 25/24 (2006.01); A61P 25/28 (2006.01); A61P 25/30 (2006.01); C07D 405/12 (2006.01)

CPC (invention and additional information)

C07D 405/12 (2013.01)

Citation (search report)

See references of WO 9962902A1

Designated contracting state (EPC)

AT BE CH DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

EPO simple patent family

WO 9962902 A1 19991209; AR 018622 A1 20011128; AU 4369599 A 19991220; BG 104988 A 20011130; BR 9910927 A 20010220; CA 2333756 A1 19991209; CN 1304408 A 20010718; CO 5021190 A1 20010327; EP 1087964 A1 20010404; GB 9811879 D0 19980729; HR P20010005 A2 20011231; HU 0102233 A2 20020529; ID 27067 A 20010222; IL 139552 D0 20020210; JP 2002517392 A 20020618; NO 20006041 A 20001129; NO 20006041 D0 20001129; PL 344594 A1 20011105; SK 17602000 A3 20010806; TR 200003569 T2 20010420

INPADOC legal status

2003-05-02 [18R] REFUSED

- Ref Legal Event Code: 18R

- Effective date: 20021205

2002-05-22 [17Q] FIRST EXAMINATION REPORT

- Ref Legal Event Code: 17Q

- Effective date: 20020411

2001-09-05 [RAP1] TRANSFER OF RIGHTS OF AN EP PUBLISHED APPLICATION

- Owner name: KNOLL GMBH

- Ref Legal Event Code: RAP1

2001-04-04 [17P] REQUEST FOR EXAMINATION FILED

- Ref Legal Event Code: 17P

- Effective date: 20001113

2001-04-04 [AK] DESIGNATED CONTRACTING STATES:

- Ref Legal Event Code: AK

- Designated State(s): AT BE CH DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

2001-04-04 [AX] REQUEST FOR EXTENSION OF THE EUROPEAN PATENT TO

- Ref Legal Event Code: AX

- Free Format Text: AL PAYMENT 20001113;LT PAYMENT 20001113;LV PAYMENT 20001113;MK PAYMENT 20001113;RO PAYMENT 20001113;SI PAYMENT 20001113