EP 1090003 A1 20010411 - 7-ALKYL- AND CYCLOALKYL-SUBSTITUTED IMIDAZOTRIAZINONES
Title (en)
7-ALKYL- AND CYCLOALKYL-SUBSTITUTED IMIDAZOTRIAZINONES
Title (de)
7-ALKYL- UND CYCLOALKYL-SUBSTITUIERTE IMIDAZOTRIAZINONE
Title (fr)
IMIDAZOTRIAZINONES A SUBSTITUTION 7-ALKYLE ET CYCLOALKYLE
Publication
Application
Priority
- DE 19827640 A 19980620
- EP 9904032 W 19990611
Abstract (en)
[origin: DE19827640A1] 2-Sulfamoylphenyl-5-alkyl-7-(cyclo)alkyl-4(3H)-imidazo(5,1-f)(1,2,4)tr iazinone derivatives (I) are new. 2-Sulfamoylphenyl-5-alkyl-7-(cyclo)alkyl-4(3H)-imidazo(5,1-f)(1,2,4)tr iazinone derivatives of formula (I) are new: R1 = 1-4C alkyl; R2 = 5-20C alkyl or 3-8C cycloalkyl; R3, R4 = H; 2-8C alkenyl; 1-10C alkyl optionally interrupted by an O atom and optionally substituted by 1-3 of CF3, OCF3, OH, halogen, COOH, benzyloxycarbonyl, 1-6C alkoxy, 2-6C alkoxycarbonyl, 1-6C alkylthio, SO3H, etc; or NR3R4 = optionally substituted optionally benzo-fused 5-7 membered heterocyclic group; or NR3R4 = a (bi)(hetero)cyclic group; and R5, R6 = H, 1-6C alkyl, OH or 1-6C alkoxy. Full definitions given in the 'Definition' section. An Independent claim is also included for the preparation of (I).
IPC 1-7
IPC 8 full level
A61K 31/53 (2006.01); A61K 31/5377 (2006.01); A61K 31/539 (2006.01); A61K 31/55 (2006.01); A61K 31/5513 (2006.01); A61K 31/675 (2006.01); A61P 7/12 (2006.01); A61P 9/00 (2006.01); A61P 9/08 (2006.01); A61P 9/10 (2006.01); A61P 15/00 (2006.01); A61P 15/10 (2006.01); A61P 21/02 (2006.01); A61P 43/00 (2006.01); C07D 487/04 (2006.01); C07D 519/00 (2006.01); C07F 9/6561 (2006.01)
CPC (source: EP US)
A61P 7/12 (2017.12 - EP); A61P 9/00 (2017.12 - EP); A61P 9/08 (2017.12 - EP); A61P 9/10 (2017.12 - EP); A61P 9/12 (2017.12 - EP); A61P 13/08 (2017.12 - EP); A61P 15/00 (2017.12 - EP); A61P 15/10 (2017.12 - EP); A61P 21/02 (2017.12 - EP); A61P 43/00 (2017.12 - EP); C07D 487/04 (2013.01 - EP US); C07F 9/6561 (2013.01 - EP US)
Citation (search report)
See references of WO 9967244A1
Designated contracting state (EPC)
DE ES FR GB IT
DOCDB simple family (publication)
DE 19827640 A1 19991223; AU 4608099 A 20000110; CA 2335193 A1 19991229; EP 1090003 A1 20010411; JP 2002518500 A 20020625; US 2005049250 A1 20050303; US 6476029 B1 20021105; US 6838459 B1 20050104; US 6943163 B2 20050913; WO 9967244 A1 19991229
DOCDB simple family (application)
DE 19827640 A 19980620; AU 4608099 A 19990611; CA 2335193 A 19990611; EP 9904032 W 19990611; EP 99929181 A 19990611; JP 2000555897 A 19990611; US 25193902 A 20020920; US 72005101 A 20010323; US 85051004 A 20040520