Global patent index - EP 1090031 A1

EP 1090031 A1 2001-04-11 - SUBSTITUTED CYCLOOCTADEPSIPEPTIDES

Title (en)

SUBSTITUTED CYCLOOCTADEPSIPEPTIDES

Title (de)

SUBSTITUIERTE CYCLOOCTADEPSIPEPTIDE

Title (fr)

CYCLOOCTADEPSIPEPTIDES SUBSTITUES

Publication

EP 1090031 A1 (DE)

Application

EP 99927953 A

Priority

  • DE 19828047 A
  • EP 9904028 W

Abstract (en)

[origin: DE19828047A1] Cyclooctadepsipeptide derivatives (I) are new. Cyclooctadepsipeptide derivatives of formula (I) are new. n = 0-2; m = 1 or 2; R<1> = SO2A in the 2- and/or 4-position; R2 = R1 or a saturated 5- or 6-membered heterocycle (which contains one N heteroatom and optionally one or two extra N or O heteroatoms, and is optionally substituted by 1-4C alkyl, (1-4C alkyl)carbonyl, (1-4C alkoxy)carbonyl or aryl, e.g. benzoyl), or an unsaturated heterocycle selected from pyrazole, imidazole, pyrrole, 1,2,4-triazole or 1,2,3-triazole, which may be substituted as before; A = NH2, mono- or di-(1-4C alkyl)amino (optionally substituted by phenyl, furyl, morpholinyl or pyridyl), bis(hydroxy-1-4C alkyl)amino, or mono- or bis(1-4C alkoxy-1-4C alkyl)amino; An Independent claim is also included for preparation of (I).

IPC 1-7 (main, further and additional classification)

C07K 11/02; A61K 38/15; C07D 273/00

IPC 8 full level (invention and additional information)

C07D 273/00 (2006.01); A61K 38/00 (2006.01); A61P 33/00 (2006.01); C07K 11/02 (2006.01)

CPC (invention and additional information)

C07K 11/02 (2013.01); A61K 38/00 (2013.01)

Citation (search report)

See references of WO 9967281A1

Designated contracting state (EPC)

AT BE CH DE DK ES FI FR GB GR IE IT LI NL PT SE

EPO simple patent family

DE 19828047 A1 19991230; AU 4511499 A 20000110; BR 9911574 A 20010320; CA 2332122 A1 19991229; CN 1307586 A 20010808; EP 1090031 A1 20010411; HU 0102476 A2 20011028; HU 0102476 A3 20030828; JP 2002518520 A 20020625; PL 345866 A1 20020114; WO 9967281 A1 19991229

INPADOC legal status

2004-07-28 [18D] DEEMED TO BE WITHDRAWN

- Ref Legal Event Code: 18D

- Effective date: 20040101

2001-04-11 [17P] REQUEST FOR EXAMINATION FILED

- Ref Legal Event Code: 17P

- Effective date: 20010124

2001-04-11 [AK] DESIGNATED CONTRACTING STATES:

- Ref Legal Event Code: AK

- Designated State(s): AT BE CH DE DK ES FI FR GB GR IE IT LI NL PT SE