Global Patent Index - EP 1093372 A1

EP 1093372 A1 20010425 - CYCLIC AMINO ACID COMPOUNDS, PHARMACEUTICAL COMPOSITIONS COMPRISING SAME, AND METHODS FOR INHIBITING $g(b)-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS BY USE OF SUCH COMPOUNDS

Title (en)

CYCLIC AMINO ACID COMPOUNDS, PHARMACEUTICAL COMPOSITIONS COMPRISING SAME, AND METHODS FOR INHIBITING $g(b)-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS BY USE OF SUCH COMPOUNDS

Title (de)

AMINOSÄUREVERBINDUNGEN, PHARMAZEUTISCHE ZUSAMMENSETZUNGEN DAMIT UND VERFAHREN ZUR HEMMUNG VON A(B)-AMYLOID-PEPTID FREISETZUNG UND/ODER DEREN SYNTHESE DURCH VERWENDUNG DIESER VERBINDUNGEN

Title (fr)

COMPOSES D'ACIDES AMINES CYCLIQUES, COMPOSITIONS PHARMACEUTIQUES LES CONTENANT ET METHODES D'INHIBITION DE LA LIBERATION DU PEPTIDE $g(b)-AMYLOIDE ET/OU DE SA SYNTHESE A L'AIDE DE CES COMPOSES

Publication

EP 1093372 A1 20010425 (EN)

Application

EP 99930600 A 19990622

Priority

  • US 9914211 W 19990622
  • US 10250798 A 19980622
  • US 16445198 A 19980930

Abstract (en)

[origin: WO9966934A1] Disclosed are compounds which inhibit beta -amyloid peptide release and/or its synthesis, and, accordingly, have utility in treating Alzheimer's disease. Also disclosed are pharmaceutical compositions comprising a compound which inhibits beta -amyloid peptide release and/or its synthesis as well as methods for treating Alzheimer's disease both prophylactically and therapeutically with such pharmaceutical compositions.

IPC 1-7

C07D 223/18; A61K 31/55; C07D 471/06; C07D 243/14; C07D 409/12; C07D 243/12; C07D 223/16; C07D 267/14; C07D 281/10; C07D 471/04; C07D 471/08; C07D 401/04; C07D 417/04; C07D 409/04; C07D 243/10; C07D 487/04; C07D 403/12; C07D 401/12

IPC 8 full level

A61K 38/00 (2006.01); A61K 31/55 (2006.01); A61P 25/28 (2006.01); A61P 43/00 (2006.01); C07D 223/14 (2006.01); C07D 223/16 (2006.01); C07D 223/18 (2006.01); C07D 243/06 (2006.01); C07D 243/10 (2006.01); C07D 243/12 (2006.01); C07D 243/14 (2006.01); C07D 243/24 (2006.01); C07D 267/02 (2006.01); C07D 267/14 (2006.01); C07D 281/02 (2006.01); C07D 281/10 (2006.01); C07D 401/04 (2006.01); C07D 401/12 (2006.01); C07D 403/12 (2006.01); C07D 409/04 (2006.01); C07D 409/12 (2006.01); C07D 417/04 (2006.01); C07D 471/04 (2006.01); C07D 471/06 (2006.01); C07D 471/08 (2006.01); C07D 487/02 (2006.01); C07D 487/04 (2006.01); C07D 487/12 (2006.01); C07D 498/02 (2006.01); C07D 513/02 (2006.01); C07K 4/00 (2006.01)

CPC (source: EP)

C07D 223/14 (2013.01); C07D 223/16 (2013.01); C07D 223/18 (2013.01); C07D 243/08 (2013.01); C07D 243/10 (2013.01); C07D 243/12 (2013.01); C07D 243/14 (2013.01); C07D 243/24 (2013.01); C07D 401/04 (2013.01); C07D 401/06 (2013.01); C07D 401/12 (2013.01); C07D 403/06 (2013.01); C07D 403/12 (2013.01); C07D 405/06 (2013.01); C07D 409/06 (2013.01); C07D 409/12 (2013.01); C07D 413/06 (2013.01); C07D 417/04 (2013.01); C07D 471/06 (2013.01); C07D 471/08 (2013.01); C07D 487/04 (2013.01); C07K 5/06026 (2013.01); A61K 38/00 (2013.01)

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

DOCDB simple family (publication)

WO 9966934 A1 19991229; AU 4710499 A 20000110; CA 2324475 A1 19991229; EP 1093372 A1 20010425; EP 1093372 A4 20040929; JP 2002518451 A 20020625

DOCDB simple family (application)

US 9914211 W 19990622; AU 4710499 A 19990622; CA 2324475 A 19990622; EP 99930600 A 19990622; JP 2000555620 A 19990622