Global Patent Index - EP 1100782 A1

EP 1100782 A1 2001-05-23 - AMINO-ALDEHYDE SOLID SUPPORT, LINKER THEREFOR AND METHODS OF PREPARATION AND USE THEREOF

Title (en)

AMINO-ALDEHYDE SOLID SUPPORT, LINKER THEREFOR AND METHODS OF PREPARATION AND USE THEREOF

Title (de)

AMINO-ALDEHYD FESTTRÄGER, LINKER DAFÜR UND VERFAHREN ZU IHRER HERSTELLUNG

Title (fr)

SUPPORT SOLIDE D'AMINO-ALDEHYDE, SA SEQUENCE DE LIAISON ET SES METHODES DE PREPARATION ET D'UTILISATION

Publication

EP 1100782 A1 (EN)

Application

EP 99938805 A

Priority

  • US 9916901 W
  • US 12200998 A

Abstract (en)

[origin: WO0005208A1] This invention provides a novel method for solid-phase peptide synthesis wherein a cyclic or linear amino aldehyde is derivatized through linkage to a solid-support, and employed in the production of biologically significant peptides, peptide derivatives, peptidomimetic compounds and analogs thereof. The method of linkage and peptide synthesis, including for combinatorial chemistry, is disclosed.

IPC 1-7 (main, further and additional classification)

C07D 211/56; A61K 31/445; C07D 401/12; C07D 405/12; C07K 1/04; C07K 17/08

IPC 8 full level (invention and additional information)

C12N 9/99 (2006.01); A61K 38/00 (2006.01); A61K 38/55 (2006.01); A61P 7/02 (2006.01); C07C 231/02 (2006.01); C07C 235/02 (2006.01); C07D 211/56 (2006.01); C07D 401/12 (2006.01); C07D 405/12 (2006.01); C07K 1/04 (2006.01); C07K 5/062 (2006.01); C08F 8/00 (2006.01); C07B 61/00 (2006.01)

CPC (invention and additional information)

C07D 401/12 (2013.01); C07D 211/56 (2013.01); C07D 405/12 (2013.01); C07K 1/045 (2013.01); C40B 40/00 (2013.01)

Citation (search report)

See references of WO 0005208A1

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

EPO simple patent family

WO 0005208 A1 20000203; WO 0005208 A9 20000803; EP 1100782 A1 20010523; JP 2002521364 A 20020716

INPADOC legal status


2005-08-03 [18D] DEEMED TO BE WITHDRAWN

- Effective date: 20050201

2001-12-05 [17Q] FIRST EXAMINATION REPORT

- Effective date: 20011023

2001-05-23 [17P] REQUEST FOR EXAMINATION FILED

- Effective date: 20010213

2001-05-23 [AK] DESIGNATED CONTRACTING STATES:

- Kind Code of Ref Document: A1

- Designated State(s): AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE