EP 1100782 A1 20010523 - AMINO-ALDEHYDE SOLID SUPPORT, LINKER THEREFOR AND METHODS OF PREPARATION AND USE THEREOF
Title (en)
AMINO-ALDEHYDE SOLID SUPPORT, LINKER THEREFOR AND METHODS OF PREPARATION AND USE THEREOF
Title (de)
AMINO-ALDEHYD FESTTRÄGER, LINKER DAFÜR UND VERFAHREN ZU IHRER HERSTELLUNG
Title (fr)
SUPPORT SOLIDE D'AMINO-ALDEHYDE, SA SEQUENCE DE LIAISON ET SES METHODES DE PREPARATION ET D'UTILISATION
Publication
Application
Priority
- US 9916901 W 19990723
- US 12200998 A 19980724
Abstract (en)
[origin: WO0005208A1] This invention provides a novel method for solid-phase peptide synthesis wherein a cyclic or linear amino aldehyde is derivatized through linkage to a solid-support, and employed in the production of biologically significant peptides, peptide derivatives, peptidomimetic compounds and analogs thereof. The method of linkage and peptide synthesis, including for combinatorial chemistry, is disclosed.
IPC 1-7
C07D 211/56; C07D 401/12; C07D 405/12; C07K 17/08; C07K 1/04; A61K 31/445
IPC 8 full level
A61K 38/00 (2006.01); A61K 38/55 (2006.01); A61P 7/02 (2006.01); C07C 231/02 (2006.01); C07C 235/02 (2006.01); C07D 211/56 (2006.01); C07D 401/12 (2006.01); C07D 405/12 (2006.01); C07K 1/04 (2006.01); C07K 5/062 (2006.01); C08F 8/00 (2006.01); C12N 9/99 (2006.01); C07B 61/00 (2006.01)
CPC (source: EP)
A61P 7/02 (2017.12); C07D 211/56 (2013.01); C07D 401/12 (2013.01); C07D 405/12 (2013.01); C07K 1/045 (2013.01); C40B 40/00 (2013.01)
Citation (search report)
See references of WO 0005208A1
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
WO 0005208 A1 20000203; WO 0005208 A9 20000803; EP 1100782 A1 20010523; JP 2002521364 A 20020716
DOCDB simple family (application)
US 9916901 W 19990723; EP 99938805 A 19990723; JP 2000561165 A 19990723