EP 1104410 A1 20010606 - NEW CARBOXYLIC ACID DERIVATIVES CARRYING KETO SIDE-CHAINS, THEIR PRODUCTION AND THEIR USE AS ENDOTHELIN-RECEPTOR ANTAGONISTS
Title (en)
NEW CARBOXYLIC ACID DERIVATIVES CARRYING KETO SIDE-CHAINS, THEIR PRODUCTION AND THEIR USE AS ENDOTHELIN-RECEPTOR ANTAGONISTS
Title (de)
NEUE CARBONSÄUREDERIVATE, DIE KETOSEITENKETTEN TRAGEN, IHRE HERSTELLUNG UND VERWENDUNG ALS ENDOTHELIN-REZEPTORANTAGONISTEN
Title (fr)
NOUVEAUX DERIVES DE L'ACIDE CARBONIQUE PORTEURS DE CHAINES LATERALES CETONE, LEUR FABRICATION ET LEUR UTILISATION COMME ANTAGONISTES DES RECEPTEURS DE L'ENDOTHELINE
Publication
Application
Priority
- DE 19836044 A 19980810
- EP 9905728 W 19990807
Abstract (en)
[origin: WO0009489A1] The invention relates to new carboxylic acid derivatives of the formula (I), where the substituents have the meaning given in the description, their production and their use as endothelin-receptor antagonists.
IPC 1-7
C07D 239/52; C07D 239/34; C07D 239/70; C07D 403/12; A61K 31/505
IPC 8 full level
A61K 31/505 (2006.01); A61K 31/517 (2006.01); A61K 31/519 (2006.01); A61K 31/53 (2006.01); A61K 45/00 (2006.01); C07D 251/22 (2006.01); A61P 9/04 (2006.01); A61P 9/10 (2006.01); A61P 9/12 (2006.01); A61P 13/08 (2006.01); A61P 13/12 (2006.01); A61P 35/00 (2006.01); A61P 43/00 (2006.01); C07D 239/34 (2006.01); C07D 239/52 (2006.01); C07D 239/60 (2006.01); C07D 239/70 (2006.01); C07D 251/52 (2006.01); C07D 401/12 (2006.01); C07D 403/12 (2006.01); C07D 405/12 (2006.01); C07D 491/048 (2006.01); C07D 495/04 (2006.01)
CPC (source: EP KR)
A61P 9/04 (2018.01 - EP); A61P 9/10 (2018.01 - EP); A61P 9/12 (2018.01 - EP); A61P 13/08 (2018.01 - EP); A61P 13/12 (2018.01 - EP); A61P 35/00 (2018.01 - EP); A61P 43/00 (2018.01 - EP); C07D 239/34 (2013.01 - EP KR); C07D 239/52 (2013.01 - EP KR); C07D 239/70 (2013.01 - EP KR); C07D 403/12 (2013.01 - EP KR)
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
WO 0009489 A1 20000224; AR 020147 A1 20020410; AU 5374199 A 20000306; BG 105236 A 20011229; BR 9912889 A 20010508; CA 2340167 A1 20000224; CN 1323298 A 20011121; CO 5261504 A1 20030331; DE 19836044 A1 20000217; EP 1104410 A1 20010606; HK 1042086 A1 20020802; HR P20010164 A2 20020430; HU P0104007 A2 20020529; HU P0104007 A3 20021228; ID 27965 A 20010503; IL 140915 A0 20020210; JP 2002522531 A 20020723; KR 20010072378 A 20010731; NO 20010622 D0 20010206; NO 20010622 L 20010206; PL 345998 A1 20020114; SK 832001 A3 20011106; TR 200100427 T2 20010723; ZA 200101975 B 20020311
DOCDB simple family (application)
EP 9905728 W 19990807; AR P990103985 A 19990810; AU 5374199 A 19990807; BG 10523601 A 20010209; BR 9912889 A 19990807; CA 2340167 A 19990807; CN 99811981 A 19990807; CO 99050715 A 19990810; DE 19836044 A 19980810; EP 99939457 A 19990807; HK 02103679 A 20020515; HR P20010164 A 20010308; HU P0104007 A 19990807; ID 20010326 A 19990807; IL 14091599 A 19990807; JP 2000564942 A 19990807; KR 20017001731 A 20010209; NO 20010622 A 20010206; PL 34599899 A 19990807; SK 832001 A 19990807; TR 200100427 T 19990807; ZA 200101975 A 20010309