EP 1119549 A4 20030129 - PROCESS FOR PREPARING 4-SUBSTITUTED-1H-INDOLE-3-GLYOXAMIDES
Title (en)
PROCESS FOR PREPARING 4-SUBSTITUTED-1H-INDOLE-3-GLYOXAMIDES
Title (de)
VERFAHREN ZUR HERSTELLUNG VON IN 4-STELLUNG SUBSTITUIERTEN 1H-INDOL-3-GLYOXAMIDEN
Title (fr)
PROCEDE DE PREPARATION DE 4-1H-INDOLE-3-GLYOXAMIDES SUBSTITUEES
Publication
Application
Priority
- US 9908325 W 19990415
- US 10360498 P 19981009
Abstract (en)
[origin: WO0021929A1] A process for preparing 1H-indole-3-glyoxamides useful for inhibiting SPLA2 and novel intermediates useful in the preparation of such compounds.
IPC 1-7
IPC 8 full level
C07D 209/22 (2006.01)
CPC (source: EP)
A61P 37/00 (2017.12); C07D 209/22 (2013.01); Y02P 20/55 (2015.11)
Citation (search report)
- [DY] EP 0675110 A1 19951004 - LILLY CO ELI [US]
- [Y] JP S6032769 A 19850219 - SAGAMI CHEM RES
- [Y] W. A. REEMERS ET AL.: "Synthesis of Indoles from 4-Oxo-4,5,6,7-tetrahydroindoles. II. Introduction of Substituents into the 4 and 5 Positions", JOURNAL OF ORGANIC CHEMISTRY., vol. 36, no. 9, 1971, AMERICAN CHEMICAL SOCIETY, WASHINGTON, DC., US, pages 1232 - 1240, XP002221421, ISSN: 0022-3263
- See references of WO 0021929A1
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
WO 0021929 A1 20000420; AR 015766 A1 20010516; AU 3564499 A 20000501; CA 2347718 A1 20000420; CO 5021230 A1 20010327; DZ 2771 A1 20031201; EP 1119549 A1 20010801; EP 1119549 A4 20030129; JP 2002527421 A 20020827; PE 20000429 A1 20000523; SV 1999000042 A 20000411; TW 472041 B 20020111
DOCDB simple family (application)
US 9908325 W 19990415; AR P990101752 A 19990415; AU 3564499 A 19990415; CA 2347718 A 19990415; CO 99022883 A 19990416; DZ 990071 A 19990414; EP 99917552 A 19990415; JP 2000575838 A 19990415; PE 00031199 A 19990415; SV 1999000042 A 19990415; TW 88106024 A 19990415