Global Patent Index - EP 1140880 A1

EP 1140880 A1 20011010 - HOMOPIPERAZINE DERIVATIVES AS SELECTIVE EMOPAMIL INHIBITORS

Title (en)

HOMOPIPERAZINE DERIVATIVES AS SELECTIVE EMOPAMIL INHIBITORS

Title (de)

HOMOPIPERAZINDERIVATE ALS SELEKTIVE EMOPAMIL-INHIBITOREN

Title (fr)

DERIVES HOMOPIPERAZINE EN TANT QU'INHIBITEURS SELECTIFS DE L'EMOPAMILE

Publication

EP 1140880 A1 20011010 (EN)

Application

EP 99962380 A 19991220

Priority

  • GB 9904330 W 19991220
  • GB 9828435 A 19981224

Abstract (en)

[origin: WO0039110A1] Homopiperazines of formula (I), wherein R<1> is hydrogen, C1-8alkyl, C2-8alkenyl or C2-8alkynyl substituted or unsubstituted with a variety of groups as defined herein; A is a ring selected from phenyl and naphthyl; R<2> at each occurrence is independently selected from a variety of groups as defined herein; m is an integer selected from the range 0 to 5 where at each occurrence R<2> is independently selected; together with processes for their manufacture and compositions containing them. Compounds of formula (I) are pharmacologically useful in the treatment of neurological disorders.

IPC 1-7

C07D 295/06; C07D 295/088; A61K 31/551; A61P 25/28; C07D 295/08; C07D 295/02; C07D 295/155; C07D 405/12

IPC 8 full level

C07D 243/08 (2006.01); A61K 31/551 (2006.01); A61P 3/10 (2006.01); A61P 9/10 (2006.01); A61P 21/02 (2006.01); A61P 25/00 (2006.01); A61P 25/16 (2006.01); A61P 25/28 (2006.01); A61P 31/18 (2006.01); C07D 295/03 (2006.01); C07D 295/073 (2006.01); C07D 295/088 (2006.01); C07D 295/096 (2006.01); C07D 295/155 (2006.01); C07D 405/12 (2006.01); C07D 295/02 (2006.01)

CPC (source: EP)

A61P 3/10 (2017.12); A61P 9/10 (2017.12); A61P 21/02 (2017.12); A61P 25/00 (2017.12); A61P 25/16 (2017.12); A61P 25/28 (2017.12); A61P 31/18 (2017.12); C07D 295/03 (2013.01); C07D 295/073 (2013.01); C07D 295/088 (2013.01); C07D 295/096 (2013.01); C07D 295/155 (2013.01); C07D 405/12 (2013.01)

Citation (search report)

See references of WO 0039110A1

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

DOCDB simple family (publication)

WO 0039110 A1 20000706; AU 1874600 A 20000731; EP 1140880 A1 20011010; GB 9828435 D0 19990217; GB 9930013 D0 20000209; JP 2002533449 A 20021008

DOCDB simple family (application)

GB 9904330 W 19991220; AU 1874600 A 19991220; EP 99962380 A 19991220; GB 9828435 A 19981224; GB 9930013 A 19991221; JP 2000591021 A 19991220