Global Patent Index - EP 1140983 A1

EP 1140983 A1 20011010 - BIS-AMINO ACID SULFONAMIDES CONTAINING N-TERMINALLY A FLUORO-SUBSTITUTED BENZYL GROUP AS HIV PROTEASE INHIBITORS

Title (en)

BIS-AMINO ACID SULFONAMIDES CONTAINING N-TERMINALLY A FLUORO-SUBSTITUTED BENZYL GROUP AS HIV PROTEASE INHIBITORS

Title (de)

BIS-AMINOSÄURE-SULFONAMIDE MIT EINER N-TERMINALEN FLUORO-SUBSTITUIERTEN BENZYLGRUPPE ALS HIV PROTEASE INHIBITORE

Title (fr)

BIS-AMINOACIDES SULFAMIDES CONTENANT UN GROUPE BENZYLE FLUORO-SUBSTITUE A L'EXTREMITE N-TERMINALE UTILISES COMME INHIBITEURS DE LA PROTEASE DU VIH

Publication

EP 1140983 A1 20011010 (EN)

Application

EP 00905604 A 20000113

Priority

  • US 0000820 W 20000113
  • US 11574699 P 19990113

Abstract (en)

[origin: WO0042060A1] This invention relates generally to bis-amino acid sulfonamides containing substituted benzyl amines of formula (I) or stereoisomeric forms, stereoisomeric mixtures, or pharmaceutically acceptable salt forms thereof, which are useful as HIV protease inhibitors, pharmaceutical compositions and diagnostic kits comprising the same, methods of using the same for treating viral infection or as assay standards or reagents, and intermediates and processes for making the same.

IPC 1-7

C07K 5/062; A61K 38/05; A61P 31/18

IPC 8 full level

A61K 31/427 (2006.01); A61K 31/472 (2006.01); A61K 31/4725 (2006.01); C12N 9/99 (2006.01); A61K 31/496 (2006.01); A61K 31/513 (2006.01); A61K 31/536 (2006.01); A61K 31/7072 (2006.01); A61K 38/00 (2006.01); A61K 45/00 (2006.01); A61P 31/18 (2006.01); A61P 43/00 (2006.01); C07K 5/06 (2006.01); C07K 5/062 (2006.01)

CPC (source: EP KR)

A61P 31/18 (2018.01 - EP); A61P 43/00 (2018.01 - EP); C07K 5/06017 (2013.01 - KR); C07K 5/06026 (2013.01 - EP); C07K 5/06191 (2013.01 - EP); A61K 38/00 (2013.01 - EP)

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

DOCDB simple family (publication)

WO 0042060 A1 20000720; AU 2725700 A 20000801; BR 0007854 A 20020115; CA 2353088 A1 20000720; CN 1336934 A 20020220; CZ 20012435 A3 20020213; EP 1140983 A1 20011010; HU P0105235 A2 20020429; HU P0105235 A3 20020828; IL 143763 A0 20020421; JP 2002536298 A 20021029; KR 20010101478 A 20011114; NO 20013338 D0 20010705; NO 20013338 L 20010913; PL 349774 A1 20020909; SK 9522001 A3 20020305; TR 200102033 T2 20011221

DOCDB simple family (application)

US 0000820 W 20000113; AU 2725700 A 20000113; BR 0007854 A 20000113; CA 2353088 A 20000113; CN 00802755 A 20000113; CZ 20012435 A 20000113; EP 00905604 A 20000113; HU P0105235 A 20000113; IL 14376300 A 20000113; JP 2000593627 A 20000113; KR 20017008803 A 20010712; NO 20013338 A 20010705; PL 34977400 A 20000113; SK 9522001 A 20000113; TR 200102033 T 20000113