EP 1144377 A4 20020502 - OXETANONE DERIVATIVES
Title (en)
OXETANONE DERIVATIVES
Title (de)
OXETANON DERIVATE
Title (fr)
DERIVES D'OXETANONE
Publication
Application
Priority
- US 0029641 W 20001027
- US 43155199 A 19991029
- US 16596099 P 19991117
- US 61832800 A 20000718
Abstract (en)
[origin: WO0132616A2] This invention relates to novel oxetanone derivative compounds and processes for producing such derivatives that are useful as lipase inhibitors. Further the invention relates to processes for producing salts and for producing pharmaceutical compositions compounds comprising at least one such oxetanone derivative or salt, as well as methods for using such compounds and compositions for inhibiting lipases.
IPC 1-7
IPC 8 full level
A61K 9/06 (2006.01); A61K 31/715 (2006.01); A61K 31/722 (2006.01); A61K 47/36 (2006.01); A61P 3/04 (2006.01); A61P 43/00 (2006.01); C07D 305/12 (2006.01); C08B 37/08 (2006.01)
CPC (source: EP)
A61K 31/715 (2013.01); A61K 31/722 (2013.01); A61P 3/04 (2017.12); A61P 43/00 (2017.12); C07D 305/12 (2013.01)
Citation (search report)
- [A] EP 0444482 A2 19910904 - HOFFMANN LA ROCHE [CH]
- [A] US 4931463 A 19900605 - BARBIER PIERRE [FR], et al
- [A] US 5175186 A 19921229 - BARBIER PIERRE [FR], et al
- [A] US 5246960 A 19930921 - BARBIER PIERRE [FR], et al
- [A] US 4983746 A 19910108 - BARBIER PIERRE [FR], et al
- [A] EP 0638317 A1 19950215 - HOFFMANN LA ROCHE [CH]
- See references of WO 0132616A2
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
WO 0132616 A2 20010510; WO 0132616 A3 20020110; AU 1238101 A 20010514; AU 1347701 A 20010514; CA 2358921 A1 20010510; CN 1342169 A 20020327; EP 1144377 A1 20011017; EP 1144377 A4 20020502; IL 144045 A0 20020421; JP 2003524685 A 20030819; MX PA01006755 A 20030515; WO 0132670 A1 20010510
DOCDB simple family (application)
US 0029641 W 20001027; AU 1238101 A 20001027; AU 1347701 A 20001027; CA 2358921 A 20001027; CN 00804391 A 20001027; EP 00973938 A 20001027; IL 14404500 A 20001027; JP 2001534769 A 20001027; MX PA01006755 A 20001027; US 0029592 W 20001027