Global Patent Index - EP 1144377 A4

EP 1144377 A4 20020502 - OXETANONE DERIVATIVES

Title (en)

OXETANONE DERIVATIVES

Title (de)

OXETANON DERIVATE

Title (fr)

DERIVES D'OXETANONE

Publication

EP 1144377 A4 20020502 (EN)

Application

EP 00973938 A 20001027

Priority

  • US 0029641 W 20001027
  • US 43155199 A 19991029
  • US 16596099 P 19991117
  • US 61832800 A 20000718

Abstract (en)

[origin: WO0132616A2] This invention relates to novel oxetanone derivative compounds and processes for producing such derivatives that are useful as lipase inhibitors. Further the invention relates to processes for producing salts and for producing pharmaceutical compositions compounds comprising at least one such oxetanone derivative or salt, as well as methods for using such compounds and compositions for inhibiting lipases.

IPC 1-7

C08B 37/08; A61K 31/715; A61P 3/04

IPC 8 full level

A61K 9/06 (2006.01); A61K 31/715 (2006.01); A61K 31/722 (2006.01); A61K 47/36 (2006.01); A61P 3/04 (2006.01); A61P 43/00 (2006.01); C07D 305/12 (2006.01); C08B 37/08 (2006.01)

CPC (source: EP)

A61K 31/715 (2013.01); A61K 31/722 (2013.01); A61P 3/04 (2017.12); A61P 43/00 (2017.12); C07D 305/12 (2013.01)

Citation (search report)

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

DOCDB simple family (publication)

WO 0132616 A2 20010510; WO 0132616 A3 20020110; AU 1238101 A 20010514; AU 1347701 A 20010514; CA 2358921 A1 20010510; CN 1342169 A 20020327; EP 1144377 A1 20011017; EP 1144377 A4 20020502; IL 144045 A0 20020421; JP 2003524685 A 20030819; MX PA01006755 A 20030515; WO 0132670 A1 20010510

DOCDB simple family (application)

US 0029641 W 20001027; AU 1238101 A 20001027; AU 1347701 A 20001027; CA 2358921 A 20001027; CN 00804391 A 20001027; EP 00973938 A 20001027; IL 14404500 A 20001027; JP 2001534769 A 20001027; MX PA01006755 A 20001027; US 0029592 W 20001027