EP 1144410 A2 20011017 - USE OF IMIDAZO 1,5-A -PYRIDO 3,2-E -PYRAZINONES AS MEDICAMENTS
Title (en)
USE OF IMIDAZO 1,5-A -PYRIDO 3,2-E -PYRAZINONES AS MEDICAMENTS
Title (de)
VERWENDUNG VON IMIDAZO¬1,5-A -PYRIDO¬3,2-E -PYRAZINONEN ALS ARZNEIMITTEL
Title (fr)
UTILISATION D'IMIDAZO 1,5-A -PYRIDO 3,2-E -PYRAZINONES COMME MEDICAMENTS
Publication
Application
Priority
- DE 19902082 A 19990120
- DE 19961302 A 19991218
- EP 0000260 W 20000114
Abstract (en)
[origin: WO0043392A2] The invention relates to the use of imidazo[1,5-a]-pyrido[3,2-e]-pyrazinones of formula (1) as inhibitors for phosphodiesterase 5 for the therapy of erectile dysfunction (impotence). The invention also relates to the use of imidazo[1,5-a]-pyrido[3,2-e]-pyrazinones of formula (1) as dual inhibitors of phosphodiesterase 3 and of phosphodiesterase 5 for the therapy of heart failure, pulmonic hypertonia and vascular diseases which are accompanied by insufficient blood supply. The invention further relates to a method for making the same.
IPC 1-7
IPC 8 full level
A61K 31/4985 (2006.01); A61P 9/04 (2006.01); A61P 9/08 (2006.01); A61P 9/10 (2006.01); A61P 9/12 (2006.01); A61P 15/10 (2006.01); A61P 43/00 (2006.01); C07D 471/14 (2006.01)
CPC (source: EP KR)
A61P 9/00 (2018.01 - EP); A61P 9/04 (2018.01 - EP); A61P 9/08 (2018.01 - EP); A61P 9/10 (2018.01 - EP); A61P 9/12 (2018.01 - EP); A61P 15/00 (2018.01 - EP); A61P 15/10 (2018.01 - EP); A61P 43/00 (2018.01 - EP); C07D 471/14 (2013.01 - EP KR)
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
Designated extension state (EPC)
MK RO SI
DOCDB simple family (publication)
WO 0043392 A2 20000727; WO 0043392 A3 20000928; AR 022318 A1 20020904; AU 2291200 A 20000807; BG 105714 A 20020228; BR 0007613 A 20011030; CA 2296224 A1 20000720; CN 1344268 A 20020410; CO 5190700 A1 20020829; CZ 20012627 A3 20020116; EA 200100792 A1 20021031; EE 200100377 A 20021015; EP 1144410 A2 20011017; HU P0105132 A2 20020529; HU P0105132 A3 20021228; ID 29790 A 20011011; IL 144156 A0 20020523; IS 5987 A 20010629; JP 2002535330 A 20021022; KR 20010101603 A 20011114; LT 2001078 A 20020826; LV 12793 A 20020220; LV 12793 B 20020520; NO 20013334 D0 20010705; NO 20013334 L 20010705; SK 10322001 A3 20020702; TR 200102121 T2 20020121
DOCDB simple family (application)
EP 0000260 W 20000114; AR P000100246 A 20000119; AU 2291200 A 20000114; BG 10571401 A 20010717; BR 0007613 A 20000114; CA 2296224 A 20000119; CN 00805307 A 20000114; CO 00002747 A 20000119; CZ 20012627 A 20000114; EA 200100792 A 20000114; EE P200100377 A 20000114; EP 00901561 A 20000114; HU P0105132 A 20000114; ID 20011592 A 20000114; IL 14415600 A 20000114; IS 5987 A 20010629; JP 2000594808 A 20000114; KR 20017009112 A 20010719; LT 2001078 A 20010719; LV 010109 A 20010719; NO 20013334 A 20010705; SK 10322001 A 20000114; TR 200102121 T 20000114