Title (en)

PYRIDOBENZODIAZEPINE AND PYRIDOBENZOXAZEPINE CARBOXYAMIDE VASOPRESSIN AGONISTS

Title (de)

PYRIDOBENZODIAZEPIN UND PYRIDOBENZOXAZEPIN CARBOXAMIDE VASOPRESSIN AGONISTEN

Title (fr)

PYRIDOBENZODIAZEPINE ET PYRIDOBENZOXAZEPINE CARBOXYAMIDE EN TANT QU'AGONISTES DE LA VASOPRESSINE

Publication

EP 1149097 A2 20011031 (EN)

Application

EP 00906916 A 20000113

Priority

• US 0000886 W 20000113
• US 24468199 A 19990204

Abstract (en)

[origin: WO0046225A2] The present invention provides benzoheterocyclic carboxyamides, particularly pyridobenzodiazepine and pyridobenzoxazepine carboxyamides, of general formula (I), wherein: W is O or NH, optionally substituted, as well as methods and pharmaceutical compositions utilizing these compounds for providing a temporary delay of urination or for the treatment of disorder which may be remedied or alleviated by vasopressin agonist activity, including diabetes insipidus, nocturnal enuresis, nocturia, urinary incontinence, bleeding or coagulation disorders.

IPC 1-7

C07D 471/04; A61K 31/551; C07D 498/04; A61K 31/553; A61P 7/12; A61P 13/00

IPC 8 full level

A61K 31/395 (2006.01); A61K 31/5513 (2006.01); A61K 31/553 (2006.01); A61P 5/10 (2006.01); A61P 7/04 (2006.01); A61P 7/12 (2006.01); A61P 13/00 (2006.01); A61P 43/00 (2006.01); C07D 471/04 (2006.01); C07D 498/04 (2006.01)

CPC (source: EP)

A61P 5/10 (2017.12); A61P 7/04 (2017.12); A61P 7/12 (2017.12); A61P 13/00 (2017.12); A61P 43/00 (2017.12); C07D 471/04 (2013.01)

Citation (search report)

See references of WO 0046225A2

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

DOCDB simple family (publication)

WO 0046225 A2 20000810; WO 0046225 A3 20001214; AU 2849600 A 20000825; CA 2358895 A1 20000810; CN 1339035 A 20020306; EP 1149097 A2 20011031; JP 2002536375 A 20021029

DOCDB simple family (application)

US 0000886 W 20000113; AU 2849600 A 20000113; CA 2358895 A 20000113; CN 00803455 A 20000113; EP 00906916 A 20000113; JP 2000597295 A 20000113