Global Patent Index - EP 1161236 A1

EP 1161236 A1 2001-12-12 - DIHYDROXY OPEN-ACID AND SALTS OF HMG-CO-A REDUCTASE INHIBITORS

Title (en)

DIHYDROXY OPEN-ACID AND SALTS OF HMG-CO-A REDUCTASE INHIBITORS

Title (de)

DIHYDROXY OFFEN-SÄURE UND SALZE VON HMG-CO-A REDUCTASE INHIBITOREN

Title (fr)

ACIDE OUVERT EN DIHYDROXY ET SELS D'INHIBITEURS DE LA HMG-CO-A REDUCTASE

Publication

EP 1161236 A1 (EN)

Application

EP 00907111 A

Priority

  • US 0002626 W
  • US 12322799 P
  • US 26474499 A

Abstract (en)

[origin: WO0053173A1] The instant invention provides methods and pharmaceutical compositions for inhibiting HMG-CoA reductase, as well as for treating and/or reducing the risk for diseases and conditions affected by inhibition of HMG-CoA reductase, comprising orally administering a therapeutically effective amount of a compound selected from a dihydroxy open acid statin and a pharmaceutically acceptable salt or ester thereof in a delayed-release pharmaceutical dosage form to a patient in need of such treatment wherein substantial release of the compound from the dosage form is delayed until after passage of the dosage form through the stomach.

IPC 1-7 (main, further and additional classification)

A61K 31/22; A61K 9/28; A61P 3/06

IPC 8 full level (invention and additional information)

A61K 9/16 (2006.01); A61K 9/28 (2006.01); A61K 9/52 (2006.01); A61K 31/194 (2006.01); A61K 31/40 (2006.01); A61K 31/4418 (2006.01); A61K 31/47 (2006.01); A61K 31/505 (2006.01); A61K 47/10 (2006.01); A61K 47/14 (2006.01); A61K 47/30 (2006.01); A61P 3/06 (2006.01); A61P 9/10 (2006.01); A61P 43/00 (2006.01)

CPC (invention and additional information)

A61K 9/2833 (2013.01)

Citation (search report)

See references of WO 0053173A1

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

EPO simple patent family

WO 0053173 A1 20000914; AR 022856 A1 20020904; AU 2866400 A 20000928; CA 2364253 A1 20000914; CO 5150193 A1 20020429; EP 1161236 A1 20011212; JP 2000256191 A 20000919; JP 2002538202 A 20021112; PE 15592000 A1 20010116; SV 2002000036 A 20020205

INPADOC legal status


2005-07-20 [18D] APPLICATION DEEMED TO BE WITHDRAWN

- Effective date: 20050118

2004-08-18 [17Q] FIRST EXAMINATION REPORT

- Effective date: 20040706

2001-12-12 [17P] REQUEST FOR EXAMINATION FILED

- Effective date: 20011008

2001-12-12 [AK] DESIGNATED CONTRACTING STATES:

- Kind Code of Ref Document: A1

- Designated State(s): AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

2001-12-12 [AX] REQUEST FOR EXTENSION OF THE EUROPEAN PATENT TO:

- Free text: AL PAYMENT 20011008;LT PAYMENT 20011008;LV PAYMENT 20011008;MK PAYMENT 20011008;RO PAYMENT 20011008;SI PAYMENT 20011008