EP 1161412 A1 20011212 - NUCLEAR RECEPTOR ARYLATING COMPOUNDS
Title (en)
NUCLEAR RECEPTOR ARYLATING COMPOUNDS
Title (de)
NUKLEARE REZEPTOREN ARYLIERENDE VERBINDUNGEN
Title (fr)
COMPOSES D'ARYLATION DE RECEPTEURS NUCLEAIRES
Publication
Application
Priority
- US 0006537 W 20000313
- US 12463599 P 19990316
Abstract (en)
[origin: WO0055118A1] The present invention discloses novel nuclear receptor ligands of formula (IA) or (IB). These compounds are useful for arylating a cysteine in a nuclear receptor.
IPC 1-7
C07C 233/66; C07C 233/65; C07C 235/38; C07K 14/705; A61P 5/00; C07D 221/14
IPC 8 full level
A61K 31/166 (2006.01); A61K 31/473 (2006.01); A61P 3/04 (2006.01); A61P 5/00 (2006.01); A61P 17/02 (2006.01); A61P 19/10 (2006.01); A61P 43/00 (2006.01); C07C 233/65 (2006.01); C07C 233/66 (2006.01); C07C 235/56 (2006.01); C07D 221/14 (2006.01)
CPC (source: EP)
A61P 3/04 (2017.12); A61P 5/00 (2017.12); A61P 17/02 (2017.12); A61P 19/10 (2017.12); A61P 43/00 (2017.12); C07C 233/65 (2013.01); C07C 233/66 (2013.01); C07C 235/56 (2013.01); C07D 221/14 (2013.01); C07C 2603/64 (2017.04)
Citation (search report)
See references of WO 0055118A1
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
WO 0055118 A1 20000921; AU 3742100 A 20001004; EP 1161412 A1 20011212; JP 2002539185 A 20021119
DOCDB simple family (application)
US 0006537 W 20000313; AU 3742100 A 20000313; EP 00916297 A 20000313; JP 2000605549 A 20000313