Global Patent Index - EP 1161412 A1

EP 1161412 A1 2001-12-12 - NUCLEAR RECEPTOR ARYLATING COMPOUNDS

Title (en)

NUCLEAR RECEPTOR ARYLATING COMPOUNDS

Title (de)

NUKLEARE REZEPTOREN ARYLIERENDE VERBINDUNGEN

Title (fr)

COMPOSES D'ARYLATION DE RECEPTEURS NUCLEAIRES

Publication

EP 1161412 A1 (EN)

Application

EP 00916297 A

Priority

  • US 0006537 W
  • US 12463599 P

Abstract (en)

[origin: WO0055118A1] The present invention discloses novel nuclear receptor ligands of formula (IA) or (IB). These compounds are useful for arylating a cysteine in a nuclear receptor.

IPC 1-7 (main, further and additional classification)

C07C 233/66; A61P 5/00; C07C 233/65; C07C 235/38; C07D 221/14; C07K 14/705

IPC 8 full level (invention and additional information)

A61K 31/166 (2006.01); A61K 31/473 (2006.01); A61P 3/04 (2006.01); A61P 5/00 (2006.01); A61P 17/02 (2006.01); A61P 19/10 (2006.01); A61P 43/00 (2006.01); C07C 233/65 (2006.01); C07C 233/66 (2006.01); C07C 235/56 (2006.01); C07D 221/14 (2006.01)

CPC (invention and additional information)

C07D 221/14 (2013.01); C07C 233/65 (2013.01); C07C 233/66 (2013.01); C07C 235/56 (2013.01); C07C 2603/64 (2017.05)

Citation (search report)

See references of WO 0055118A1

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

EPO simple patent family

WO 0055118 A1 20000921; AU 3742100 A 20001004; EP 1161412 A1 20011212; JP 2002539185 A 20021119

INPADOC legal status


2004-01-02 [18D] DEEMED TO BE WITHDRAWN

- Effective date: 20030617

2003-03-26 [17Q] FIRST EXAMINATION REPORT

- Effective date: 20030206

2001-12-12 [17P] REQUEST FOR EXAMINATION FILED

- Effective date: 20010907

2001-12-12 [AK] DESIGNATED CONTRACTING STATES:

- Kind Code of Ref Document: A1

- Designated State(s): AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

2001-12-12 [AX] REQUEST FOR EXTENSION OF THE EUROPEAN PATENT TO

- Free text: AL;LT;LV;MK;RO;SI