EP 1161431 A4 20020424 - 6-AZAINDOLE COMPOUNDS AS ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE
Title (en)
6-AZAINDOLE COMPOUNDS AS ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE
Title (de)
6-AZAINDOL-VERBINDUNGEN ALS ANTAGONISTEN DES GONADOTROPIN-FREISETZUNGS HORMONES
Title (fr)
COMPOSES 6-AZAINDOLE UTILISES COMME ANTAGONISTES D'UNE HORMONE LIBERANT LA GONADOTROPINE
Publication
Application
Priority
- US 0005799 W 20000306
- US 12362099 P 19990310
Abstract (en)
[origin: WO0053602A1] There are disclosed compounds of formula (I) and pharmaceutically acceptable salts thereof which are useful as antagonists of GnRH and as such may be useful for the treatment of a variety of sex-hormone related and other conditions in both men and women.
IPC 1-7
C07D 471/04; C07D 471/08; C07D 401/06; C07D 401/12; A61K 31/44; A61K 31/435; A61P 15/00
IPC 8 full level
A61K 31/437 (2006.01); A61K 31/439 (2006.01); A61K 38/00 (2006.01); A61K 38/04 (2006.01); A61K 38/22 (2006.01); A61K 45/06 (2006.01); A61P 1/00 (2006.01); A61P 5/04 (2006.01); A61P 15/18 (2006.01); A61P 17/00 (2006.01); A61P 25/00 (2006.01); A61P 35/00 (2006.01); A61P 37/00 (2006.01); C07D 519/00 (2006.01)
CPC (source: EP)
A61K 45/06 (2013.01); A61P 1/00 (2017.12); A61P 5/04 (2017.12); A61P 15/00 (2017.12); A61P 15/18 (2017.12); A61P 17/00 (2017.12); A61P 25/00 (2017.12); A61P 35/00 (2017.12); A61P 37/00 (2017.12); C07D 519/00 (2013.01)
Citation (search report)
- [Y] US 5756507 A 19980526 - GOULET MARK [US], et al
- [Y] US 5780437 A 19980714 - GOULET MARK [US], et al
- [Y] WO 9721703 A1 19970619 - MERCK & CO INC [US], et al
- [Y] WO 9721707 A1 19970619 - MERCK & CO INC [US], et al
- See references of WO 0053602A1
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
WO 0053602 A1 20000914; AU 3868500 A 20000928; CA 2366615 A1 20000914; EP 1161431 A1 20011212; EP 1161431 A4 20020424; JP 2002539124 A 20021119
DOCDB simple family (application)
US 0005799 W 20000306; AU 3868500 A 20000306; CA 2366615 A 20000306; EP 00917757 A 20000306; JP 2000604039 A 20000306