Global Patent Index - EP 1165076 A4

EP 1165076 A4 20020515 - 6-AZAINDOLE COMPOUNDS AS ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE

Title (en)

6-AZAINDOLE COMPOUNDS AS ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE

Title (de)

6-AZAINDOLVERBINDUNGEN ALS ANTAGONISTEN DES GONADOLIBERINS

Title (fr)

COMPOSES DE 6-AZAINDOLE COMME ANTAGONISTES DE LA GONADOLIBERINE

Publication

EP 1165076 A4 20020515 (EN)

Application

EP 00912193 A 20000306

Priority

  • US 0005933 W 20000306
  • US 12364099 P 19990310

Abstract (en)

[origin: WO0053181A1] There are disclosed compounds of formula (I) and pharmaceutically acceptable salts thereof which are useful as antagonists of GnRH and as such may be useful for the treatment of a variety of sex-hormone related and other conditions in both men and women.

IPC 1-7

A61K 31/437; A61K 31/435; A61K 31/495; A61K 31/497; A61K 31/498; A61K 31/506; A61K 31/517; A61K 31/541; A61K 31/5355; A61P 5/04; C07D 519/00; C07D 471/04

IPC 8 full level

A61K 31/437 (2006.01); A61P 5/04 (2006.01); C07D 453/06 (2006.01); C07D 471/04 (2006.01); C07D 519/00 (2006.01)

CPC (source: EP)

A61K 31/437 (2013.01); A61P 1/00 (2017.12); A61P 5/02 (2017.12); A61P 5/04 (2017.12); A61P 5/24 (2017.12); A61P 15/00 (2017.12); A61P 15/18 (2017.12); A61P 17/00 (2017.12); A61P 25/20 (2017.12); A61P 35/00 (2017.12); A61P 37/02 (2017.12); C07D 453/06 (2013.01); C07D 471/04 (2013.01)

Citation (search report)

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

DOCDB simple family (publication)

WO 0053181 A1 20000914; AU 3396000 A 20000928; CA 2367126 A1 20000914; EP 1165076 A1 20020102; EP 1165076 A4 20020515; JP 2002538206 A 20021112

DOCDB simple family (application)

US 0005933 W 20000306; AU 3396000 A 20000306; CA 2367126 A 20000306; EP 00912193 A 20000306; JP 2000603670 A 20000306