EP 1165076 A4 20020515 - 6-AZAINDOLE COMPOUNDS AS ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE
Title (en)
6-AZAINDOLE COMPOUNDS AS ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE
Title (de)
6-AZAINDOLVERBINDUNGEN ALS ANTAGONISTEN DES GONADOLIBERINS
Title (fr)
COMPOSES DE 6-AZAINDOLE COMME ANTAGONISTES DE LA GONADOLIBERINE
Publication
Application
Priority
- US 0005933 W 20000306
- US 12364099 P 19990310
Abstract (en)
[origin: WO0053181A1] There are disclosed compounds of formula (I) and pharmaceutically acceptable salts thereof which are useful as antagonists of GnRH and as such may be useful for the treatment of a variety of sex-hormone related and other conditions in both men and women.
IPC 1-7
A61K 31/437; A61K 31/435; A61K 31/495; A61K 31/497; A61K 31/498; A61K 31/506; A61K 31/517; A61K 31/541; A61K 31/5355; A61P 5/04; C07D 519/00; C07D 471/04
IPC 8 full level
A61K 31/437 (2006.01); A61P 5/04 (2006.01); C07D 453/06 (2006.01); C07D 471/04 (2006.01); C07D 519/00 (2006.01)
CPC (source: EP)
A61K 31/437 (2013.01); A61P 1/00 (2017.12); A61P 5/02 (2017.12); A61P 5/04 (2017.12); A61P 5/24 (2017.12); A61P 15/00 (2017.12); A61P 15/18 (2017.12); A61P 17/00 (2017.12); A61P 25/20 (2017.12); A61P 35/00 (2017.12); A61P 37/02 (2017.12); C07D 453/06 (2013.01); C07D 471/04 (2013.01)
Citation (search report)
- [AD] US 5780437 A 19980714 - GOULET MARK [US], et al
- [AD] US 5849764 A 19981215 - GOULET MARK [US], et al
- See references of WO 0053181A1
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
WO 0053181 A1 20000914; AU 3396000 A 20000928; CA 2367126 A1 20000914; EP 1165076 A1 20020102; EP 1165076 A4 20020515; JP 2002538206 A 20021112
DOCDB simple family (application)
US 0005933 W 20000306; AU 3396000 A 20000306; CA 2367126 A 20000306; EP 00912193 A 20000306; JP 2000603670 A 20000306