Global Patent Index - EP 1165575 A1

EP 1165575 A1 20020102 - PHOSPHATE CONTAINING MACROCYCLIC IMMUNOMODULATORS

Title (en)

PHOSPHATE CONTAINING MACROCYCLIC IMMUNOMODULATORS

Title (de)

PHOSPHAT-ENTHALTENDE MAKROZYCLISCHE IMMUNOMODULATOREN

Title (fr)

PHOSPHATE CONTENANT DES IMMUNOMODULATEURS MACROCYCLIQUES

Publication

EP 1165575 A1 20020102 (EN)

Application

EP 00918274 A 20000323

Priority

  • US 0007639 W 20000323
  • US 28313199 A 19990331

Abstract (en)

[origin: WO0058318A1] The present invention relates to novel compounds of formula (I) which are useful as immunomodulators, in particular, macrolide immunosuppressants. The invention also relates to the preparation of compounds of formula (I), compositions containing such compounds, and methods of using such compounds.

IPC 1-7

C07F 9/6561; A61K 31/675; A61P 37/06

IPC 8 full level

A61K 31/661 (2006.01); A61P 17/00 (2006.01); A61P 17/02 (2006.01); A61P 17/06 (2006.01); A61P 17/10 (2006.01); A61P 17/14 (2006.01); A61P 37/00 (2006.01); A61P 37/06 (2006.01); C07F 9/6561 (2006.01)

CPC (source: EP)

A61P 17/00 (2017.12); A61P 17/02 (2017.12); A61P 17/06 (2017.12); A61P 17/10 (2017.12); A61P 17/14 (2017.12); A61P 37/00 (2017.12); A61P 37/06 (2017.12); C07F 9/6561 (2013.01)

Citation (search report)

See references of WO 0058318A1

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

DOCDB simple family (publication)

WO 0058318 A1 20001005; CA 2368463 A1 20001005; EP 1165575 A1 20020102; JP 2002540211 A 20021126; MX PA01009935 A 20020506

DOCDB simple family (application)

US 0007639 W 20000323; CA 2368463 A 20000323; EP 00918274 A 20000323; JP 2000608018 A 20000323; MX PA01009935 A 20000323